SCHEMBL2931406

SCHEMBL2931406

NC[C@@H]1[C@@H]2C[C@@H]2CN1C(=O)c1ccccc1-c1cccc(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 8/20 0.48
HCRTR2 O43614 7/20 0.48
CHRM1 P11229 8/20 0.42
CHRM3 P20309 6/20 0.42
CHRM2 P08172 2/20 0.42
CHRM4 P08173 2/20 0.42
RORC P51449 1/20 0.36
RORB Q92753 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3415866 1.00 HCRTR1 (0.48) HCRTR1HCRTR2CHRM1CHRM3CHRM2
SCHEMBL2924532 0.88 SLC6A4 (0.40) HCRTR1HCRTR2
SCHEMBL2930272 0.88 CHRM1 (0.46) HCRTR1HCRTR2CHRM1CHRM3RORC
SCHEMBL2929614 0.88 CHRM1 (0.46) HCRTR1HCRTR2CHRM1
SCHEMBL3415643 0.88 HCRTR1 (0.46) HCRTR1HCRTR2
SCHEMBL2930541 0.88 HCRTR1 (0.46) HCRTR1HCRTR2
SCHEMBL2926961 0.87 MEN1 (0.43) HCRTR1HCRTR2CHRM3
SCHEMBL3414068 0.87 MEN1 (0.43) HCRTR1HCRTR2CHRM3
SCHEMBL3416000 0.87 HCRTR1 (0.50) HCRTR1HCRTR2CHRM3
SCHEMBL2930074 0.85 SLC6A7 (0.35) HCRTR1HCRTR2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079690-B1 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-09-15 EP claimed
EP-2079690-B1 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-09-15 EP disclosed