SCHEMBL29314115

SCHEMBL29314115

CCCC[C@@H](CC)Nc1ncc(C#N)c(NCCOC)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.36
CTSK P43235 1/20 0.35
ALDH1A1 P00352 4/20 0.35
HPGD P15428 2/20 0.35
ALOX12 P18054 1/20 0.35
HTT P42858 1/20 0.35
ATM Q13315 1/20 0.35
PLK1 P53350 1/20 0.35
FGFR4 P22455 4/20 0.35
POLB P06746 1/20 0.34
LRRK2 Q5S007 4/20 0.34
KDM4E B2RXH2 4/20 0.34
SIRT5 Q9NXA8 1/20 0.34
MEN1 O00255 1/20 0.33
GAA P10253 1/20 0.33
KMT2A Q03164 1/20 0.33
PKM P14618 1/20 0.33
JAK2 O60674 1/20 0.33
JAK3 P52333 1/20 0.33
CDK5 Q00535 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4578984 0.77 CTSK (0.42) CHEK1CTSKALDH1A1HPGDALOX12
SCHEMBL29316281 0.76 LRRK2 (0.40) PLK1LRRK2JAK2JAK3
SCHEMBL29313602 0.71 POLB (0.48) ALDH1A1HPGDPOLBKDM4ESIRT5
SCHEMBL4579364 0.71 SMN1; SMN2 (0.45) CTSKALDH1A1HPGDALOX12HTT
SCHEMBL23019442 0.68 LRRK2 (0.36) PLK1LRRK2
SCHEMBL11160250 0.67 MAPT (0.47) ALDH1A1HPGDFGFR4KDM4EMEN1
SCHEMBL29313990 0.66 CHEK1 (0.40) CHEK1PLK1LRRK2JAK2JAK3
SCHEMBL4768640 0.65 POLB (0.49) ALDH1A1HPGDHTTPOLBLRRK2
SCHEMBL23019450 0.65 PLK1 (0.40) PLK1FGFR4LRRK2
SCHEMBL29313687 0.65 POLB (0.41) CHEK1ALDH1A1HPGDPOLBLRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3782986-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2024-07-10 EP disclosed