SCHEMBL29314732

SCHEMBL29314732

CNc1ncc(C#N)c(-c2ccc(S(N)(=O)=O)cc2)n1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 6/20 0.61
CDK1 P06493 6/20 0.61
CCNT1 O60563 3/20 0.57
CCNA2 P20248 3/20 0.57
CDK2 P24941 3/20 0.57
CDK9 P50750 3/20 0.57
CCNA1 P78396 2/20 0.57
CHUK O15111 4/20 0.51
IKBKB O14920 4/20 0.50
CCNB1 P14635 2/20 0.48
CDK7 P50613 2/20 0.48
CCNH P51946 2/20 0.48
CA1 P00915 3/20 0.46
CA2 P00918 3/20 0.46
CA9 Q16790 3/20 0.46
CA12 O43570 2/20 0.46
CA4 P22748 1/20 0.46
CA6 P23280 1/20 0.46
CA5A P35218 1/20 0.46
CA7 P43166 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24477853 0.81 KDR (0.76) KDRCDK1CCNT1CCNA2CDK2
SCHEMBL24478147 0.80 KDR (0.74) KDRCDK1CCNT1CCNA2CDK2
SCHEMBL24478142 0.79 CCNT1 (0.62) KDRCDK1CCNT1CCNA2CDK2
SCHEMBL24478141 0.75 CDK1 (0.62) KDRCDK1CCNT1CCNA2CDK2
SCHEMBL29315373 0.75 KDR (0.48) KDRCDK1CCNT1CCNA2CDK2
SCHEMBL1593001 0.73 CCNT1 (1.00) CDK1CCNT1CCNA2CDK2CDK9
SCHEMBL29314862 0.73 ADORA1 (0.64) KDRCDK1ADORA2AADORA1
SCHEMBL24478143 0.73 CDK1 (0.62) KDRCDK1CCNT1CCNA2CDK2
SCHEMBL24478139 0.73 KDR (0.64) KDRCDK1CCNT1CCNA2CDK2
SCHEMBL6221829 0.71 NPC1 (0.67) KDRCDK1CCNT1CCNA2CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3782986-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2024-07-10 EP disclosed