SCHEMBL29314862

SCHEMBL29314862

CNc1ncc(C#N)c(-c2cccnc2)n1

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 6/20 0.64
KDR P35968 9/20 0.57
CDK1 P06493 6/20 0.54
ADORA2A P29274 5/20 0.50
ADORA2B P29275 1/20 0.50
ALDH1A1 P00352 2/20 0.44
ALOX15 P16050 1/20 0.44
RAB9A P51151 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CNR1 P21554 1/20 0.43
CNR2 P34972 1/20 0.43
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
HPGD P15428 1/20 0.42
CLK1 P49759 1/20 0.42
AXL P30530 1/20 0.42
TYRO3 Q06418 1/20 0.42
MERTK Q12866 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29315373 0.82 KDR (0.48) ADORA1KDRCDK1ADORA2AALDH1A1
SCHEMBL29314691 0.78 ADORA1 (0.63) ADORA1KDRCDK1ADORA2AADORA2B
SCHEMBL20764165 0.78 ADORA1 (0.53) ADORA1KDRCDK1ADORA2AADORA2B
SCHEMBL6033927 0.75 KDR (0.61) KDRCDK1ADORA2AADORA2B
SCHEMBL29314718 0.75 CYP11B1 (0.48) ADORA1KDRCDK1ADORA2AALDH1A1
SCHEMBL6034180 0.74 KDR (0.56) KDRCDK1
SCHEMBL6034534 0.74 MAPK10 (0.55) ADORA1KDRCDK1ADORA2AADORA2B
SCHEMBL29314783 0.74 KDR (0.47) ADORA1KDRCDK1ADORA2AADORA2B
SCHEMBL29314680 0.74 KDR (0.45) ADORA1KDRCDK1ADORA2AADORA2B
SCHEMBL29314732 0.73 KDR (0.61) ADORA1KDRCDK1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3782986-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2024-07-10 EP disclosed