SCHEMBL29314924

SCHEMBL29314924

CP(C)(=O)c1ccc(-c2cnc3nnn(C(Cl)c4ccc5ncccc5c4)c3n2)cc1F

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MET P08581 20/20 0.52
PDE4C Q08493 3/20 0.52
PDE4D Q08499 3/20 0.52
PDE3B Q13370 3/20 0.52
PDE3A Q14432 3/20 0.52
PDE1A P54750 1/20 0.40
PDE1C Q14123 1/20 0.40
PDE11A Q9HCR9 1/20 0.40
PDE10A Q9Y233 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22109364 0.91 MET (0.64) METPDE4CPDE4DPDE3BPDE3A
SCHEMBL29314877 0.87 MET (0.56) METPDE4CPDE4DPDE3BPDE3A
SCHEMBL29314899 0.84 MET (0.48) METPDE4CPDE4DPDE3BPDE3A
SCHEMBL29314897 0.82 MET (0.54) METPDE4CPDE4DPDE3BPDE3A
SCHEMBL22109177 0.81 MET (0.47) METPDE4CPDE4DPDE3BPDE3A
SCHEMBL30948864 0.80 MET (0.71) METPDE3BPDE3APDE10A
SCHEMBL22109410 0.80 MET (0.71) METPDE3BPDE3APDE10A
SCHEMBL29315005 0.80 MET (0.46) METPDE4CPDE4DPDE3BPDE3A
SCHEMBL30948872 0.80 MET (0.71) METPDE3BPDE3APDE10A
SCHEMBL29314878 0.79 MET (0.49) METPDE4CPDE4DPDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3893872-B1 ORGANOPHOSPHORUS-SUBSTITUTED COMPOUNDS AS C-MET INHIBITORS AND THERAPEUTIC USES THEREOF BETA PHARMA INC (US) 2024-07-17 EP disclosed