SCHEMBL29315239

SCHEMBL29315239

CNc1ncc(C#N)c(-c2c[nH]nc2C)n1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 1/20 0.42
CCNT1 O60563 14/20 0.41
CCNA2 P20248 14/20 0.41
CDK2 P24941 14/20 0.41
CDK9 P50750 14/20 0.41
CCNA1 P78396 8/20 0.41
CDK1 P06493 9/20 0.39
KDR P35968 5/20 0.39
CCNB1 P14635 5/20 0.37
CDK7 P50613 5/20 0.37
CCNH P51946 5/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29314750 0.82 HSP90AB1 (0.39) HSP90AB1CCNT1CCNA2CDK2CDK9
SCHEMBL22998096 0.78 HSP90AB1 (0.41) HSP90AB1
SCHEMBL13523666 0.74 KDM4E (0.41) CCNT1CCNA2CDK2CDK9CCNA1
SCHEMBL23019360 0.74 KDR (0.41) HSP90AB1CCNT1CCNA2CDK2CDK9
SCHEMBL21410027 0.73 HSP90AB1 (0.38) HSP90AB1
SCHEMBL21549440 0.72 CDK7 (0.57) CCNT1CDK2CDK9CDK1KDR
SCHEMBL22684859 0.70 CCNT1 (0.54) CCNT1CCNA2CDK2CDK9CCNA1
SCHEMBL29315387 0.70 KDR (0.37) HSP90AB1CCNT1CCNA2CDK2CDK9
SCHEMBL29314779 0.70 BRD4 (0.42) CCNT1CCNA2CDK2CDK9CCNA1
SCHEMBL29314680 0.70 KDR (0.45) CCNT1CCNA2CDK2CDK9CCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3782986-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2024-07-10 EP disclosed