SCHEMBL29314680

SCHEMBL29314680

CNc1ncc(C#N)c(-c2cccnc2OC)n1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDR P35968 6/20 0.45
CDK1 P06493 4/20 0.45
IDH1 O75874 1/20 0.40
ADORA1 P30542 6/20 0.38
NAAA Q02083 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
ADORA2A P29274 3/20 0.37
ADORA2B P29275 1/20 0.37
CCNT1 O60563 2/20 0.36
CCNA2 P20248 2/20 0.36
CDK2 P24941 2/20 0.36
CDK9 P50750 2/20 0.36
CCNA1 P78396 2/20 0.36
PIK3CA P42336 1/20 0.36
BTK Q06187 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25597187 0.76 IDH1 (0.45) KDRCDK1IDH1
SCHEMBL29314862 0.74 ADORA1 (0.64) KDRCDK1ADORA1ADORA2AADORA2B
SCHEMBL29314783 0.72 KDR (0.47) KDRCDK1ADORA1ADORA2AADORA2B
SCHEMBL3613255 0.72 TEK (0.51) KDRIDH1
SCHEMBL20406383 0.70 PDE10A (0.46) PIK3CABTK
SCHEMBL29315239 0.70 HSP90AB1 (0.42) KDRCDK1CCNT1CCNA2CDK2
SCHEMBL564719 0.70 GRM5 (0.49) L3MBTL1
SCHEMBL29530525 0.70 GRM5 (0.49) L3MBTL1
SCHEMBL21549440 0.69 CDK7 (0.57) KDRCDK1CCNT1CDK2CDK9
SCHEMBL23019360 0.69 KDR (0.41) KDRCDK1ADORA1ADORA2ACCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3782986-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2024-07-10 EP disclosed