SCHEMBL29315908

SCHEMBL29315908

CCc1ncc(C#N)c(NC2COC2)n1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 4/20 0.40
IRAK4 Q9NWZ3 6/20 0.34
MBOAT4 Q96T53 3/20 0.33
PRKCQ Q04759 2/20 0.33
PRKCD Q05655 2/20 0.33
ALDH1A1 P00352 2/20 0.33
ACHE P22303 1/20 0.33
KDM4E B2RXH2 1/20 0.32
HPGD P15428 1/20 0.32
ATM Q13315 1/20 0.32
HIF1A Q16665 1/20 0.32
PGK1 P00558 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
HRH1 P35367 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29315748 0.90 LRRK2 (0.39) LRRK2IRAK4MBOAT4PRKCQPRKCD
SCHEMBL29315949 0.80 LRRK2 (0.48) LRRK2IRAK4PRKCQPRKCDCYP2C9
SCHEMBL30662127 0.79 CSNK1A1 (0.45) LRRK2IRAK4ALDH1A1ACHE
SCHEMBL21409882 0.79 CSNK1A1 (0.45) LRRK2IRAK4ALDH1A1ACHE
SCHEMBL8595874 0.77 ACHE (0.42) LRRK2MBOAT4PRKCQPRKCDACHE
SCHEMBL29316281 0.74 LRRK2 (0.40) LRRK2IRAK4PRKCQPRKCDCYP2C9
SCHEMBL21066963 0.68 PRKCQ (0.39) LRRK2PRKCQALDH1A1ACHE
SCHEMBL13736333 0.68 NPSR1 (0.44) LRRK2PRKCQALDH1A1KDM4EHPGD
SCHEMBL14657063 0.68 LRRK2 (0.50) LRRK2IRAK4PRKCQPRKCDCYP2C9
SCHEMBL21162418 0.68 LRRK2 (0.50) LRRK2IRAK4PRKCQPRKCDCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3782986-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2024-07-10 EP disclosed