SCHEMBL2932064

SCHEMBL2932064

NC(=O)Nc1sc(-c2ccc(CN3CCCC(CO)C3)cc2)cc1OC(N)=O

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 9/20 0.54
CYP2D6 P10635 1/20 0.49
ACKR3 P25106 1/20 0.42
MAP3K7 O43318 1/20 0.41
MAPT P10636 1/20 0.41
LTA4H P09960 1/20 0.40
IKBKB O14920 3/20 0.40
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
MAOB P27338 1/20 0.39
S1PR1 P21453 1/20 0.39
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2932338 0.89 CHEK1 (0.55) CHEK1MAP3K7IKBKBACHE
SCHEMBL2930060 0.87 CHEK1 (0.70) CHEK1MAP3K7MAPTIKBKBALDH1A1
SCHEMBL1927365 0.86 CHEK1 (0.73) CHEK1CYP2D6MAPTIKBKB
SCHEMBL2933445 0.86 CHEK1 (0.72) CHEK1CYP2D6MAP3K7MAPTIKBKB
SCHEMBL2933338 0.85 CHEK1 (0.52) CHEK1MAP3K7IKBKB
SCHEMBL2926946 0.83 KDM4E (0.53) CHEK1MAPTALDH1A1POLB
SCHEMBL2932566 0.83 CHEK1 (0.57) CHEK1CYP2D6MAP3K7IKBKBALDH1A1
SCHEMBL2931062 0.81 CHEK1 (0.59) CHEK1MAP3K7IKBKBALDH1A1
SCHEMBL2933039 0.80 CHEK1 (0.73) CHEK1MAP3K7IKBKB
SCHEMBL6646218 0.80 CYP2D6 (0.56) CHEK1CYP2D6ACKR3MAP3K7MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1421074-B1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2010-09-29 EP claimed