SCHEMBL2932065

SCHEMBL2932065

O=C(O)N(F)c1ccc(Oc2ccnc3[nH]c(=O)cnc23)cc1

nearest known ligand 0.52

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BRAF P15056 20/20 0.52
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2935570 0.87 BRAF (0.48) BRAFKCNH2
SCHEMBL3757658 0.85 BRAF (0.50) BRAFKCNH2
SCHEMBL2937399 0.84 BRAF (0.48) BRAFKCNH2
SCHEMBL2928516 0.82 BRAF (0.52) BRAF
SCHEMBL9909763 0.80 BRAF (0.53) BRAF
SCHEMBL2930178 0.80 BRAF (0.63) BRAFKCNH2
SCHEMBL12455757 0.78 BRAF (0.52) BRAF
SCHEMBL15925262 0.77 BRAF (0.62) BRAF
SCHEMBL3751698 0.75 BRAF (0.47) BRAFKCNH2
SCHEMBL28690834 0.75 BRAF (0.68) BRAFKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229391-A1 PYRIDO[2,3-B]PYRAZINE-8-SUBSTITUTED COMPOUNDS AND THEIR USE Cancer Research Technology Limited (GB) 2010-09-22 EP disclosed
WO-2009077766-A1 PYRIDO[2,3-B]PYRAZINE-8-SUBSTITUTED COMPOUNDS AND THEIR USE CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2009-06-25 WO disclosed