SCHEMBL29324454

SCHEMBL29324454

CNCCn1cc(C(=O)NCc2cccc(C)n2)c(=O)c2cc3c(cc21)OC(F)(F)O3

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.41
ALDH1A1 P00352 6/20 0.41
MEN1 O00255 4/20 0.41
MAPK1 P28482 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KDM4E B2RXH2 2/20 0.41
PDE4A P27815 4/20 0.40
PDE4B Q07343 4/20 0.40
PDE4C Q08493 4/20 0.40
PDE4D Q08499 4/20 0.40
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
USP2 O75604 2/20 0.38
HPGD P15428 2/20 0.38
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38
YWHAG P61981 1/20 0.38
POLR1A O95602 1/20 0.38
CNR2 P34972 1/20 0.37
ADORA3 P0DMS8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29324439 0.91 ALDH1A1 (0.43) KMT2AALDH1A1MEN1MAPK1NPSR1
SCHEMBL29324080 0.89 POLR1A (0.40) KMT2AALDH1A1MEN1MAPK1NPSR1
SCHEMBL31103594 0.82 ALDH1A1 (0.36) KMT2AALDH1A1MEN1MAPK1NPSR1
SCHEMBL29324385 0.80 PDE4A (0.50) KMT2AALDH1A1MEN1MAPK1NPSR1
SCHEMBL31103664 0.79 KMT2A (0.38) KMT2AALDH1A1MEN1MAPK1NPSR1
SCHEMBL29324375 0.78 PDE4A (0.47) KMT2AALDH1A1MEN1MAPK1NPSR1
SCHEMBL29324423 0.77 KMT2A (0.48) KMT2AALDH1A1MEN1KDM4EHSD17B10
SCHEMBL31103663 0.72 PDE4A (0.44) KMT2AALDH1A1MEN1KDM4EPDE4A
SCHEMBL29324061 0.72 PDE4A (0.44) KMT2AALDH1A1MEN1KDM4EPDE4A
SCHEMBL31103631 0.70 PDE4A (0.41) KMT2AALDH1A1MEN1MAPK1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024151425-A1 COMPOUNDS AND METHOD FOR TREATING HIV INFECTION THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2024-07-18 WO disclosed