SCHEMBL2933193

SCHEMBL2933193

Cc1cc(C(=O)N2CCCOc3ccccc32)ccc1CN

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 10/20 0.59
POLB P06746 1/20 0.50
NR3C2 P08235 1/20 0.47
ALDH1A1 P00352 2/20 0.47
TSHR P16473 2/20 0.47
USP2 O75604 1/20 0.47
LMNA P02545 1/20 0.47
NOTUM Q6P988 1/20 0.44
MAPT P10636 1/20 0.44
THRB P10828 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2704087 0.88 ALDH1A1 (0.50) AVPR2ALDH1A1TSHRUSP2LMNA
SCHEMBL2705045 0.86 AVPR2 (0.47) AVPR2POLBALDH1A1TSHRUSP2
SCHEMBL2933189 0.84 AVPR2 (0.52) AVPR2POLBNR3C2ALDH1A1TSHR
SCHEMBL1346004 0.80 AVPR2 (0.69) AVPR2
Hydrochloric Acid SCHEMBL4195564 0.79 AVPR2 (0.68) AVPR2
SCHEMBL5230382 0.78 AVPR2 (0.57) AVPR2NOTUM
Hydrochloric Acid SCHEMBL5235888 0.78 AVPR2 (0.47) AVPR2
SCHEMBL7353012 0.78 POLB (0.64) AVPR2POLBNR3C2ALDH1A1TSHR
Hydrochloric Acid SCHEMBL5270039 0.77 AVPR2 (0.56) AVPR2
SCHEMBL2938323 0.77 AVPR2 (0.46) AVPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1778677-B1 HETEROCYCLIC CONDENSED COMPOUNDS USEFUL AS ANTIDIURETIC AGENTS VANTIA LTD (GB) 2010-02-03 EP claimed