SCHEMBL2933189

SCHEMBL2933189

Cc1cc(C(=O)N2CCCOc3ccccc32)ccc1C(N)=O

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 2/20 0.52
POLB P06746 1/20 0.52
NR3C2 P08235 2/20 0.48
NOTUM Q6P988 1/20 0.46
ALDH1A1 P00352 2/20 0.46
TSHR P16473 2/20 0.46
USP2 O75604 1/20 0.46
LMNA P02545 1/20 0.46
CTSD P07339 1/20 0.43
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
GRM7 Q14831 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2704086 0.88 ALDH1A1 (0.49) AVPR2POLBALDH1A1TSHRUSP2
SCHEMBL2705044 0.86 AVPR2 (0.47) AVPR2POLBALDH1A1TSHRHDAC1
SCHEMBL2933193 0.84 AVPR2 (0.59) AVPR2POLBNR3C2NOTUMALDH1A1
SCHEMBL7353012 0.79 POLB (0.64) AVPR2POLBNR3C2NOTUMALDH1A1
SCHEMBL7012627 0.79 PDE4A (0.53) AVPR2POLBNR3C2NOTUMALDH1A1
SCHEMBL2937767 0.79 AVPR2 (0.64) AVPR2PDE4APDE4BPDE4CPDE4D
SCHEMBL7017182 0.78 PDE4A (0.52) AVPR2POLBNR3C2NOTUMALDH1A1
SCHEMBL7347470 0.76 AVPR1A (0.68) AVPR2
SCHEMBL19859267 0.76 NOTUM (0.58) POLBNOTUMTSHRLMNAHDAC1
SCHEMBL4901707 0.76 POLB (0.62) AVPR2POLBNR3C2NOTUMLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1778677-B1 HETEROCYCLIC CONDENSED COMPOUNDS USEFUL AS ANTIDIURETIC AGENTS VANTIA LTD (GB) 2010-02-03 EP claimed