SCHEMBL293326

SCHEMBL293326

N[C@@H]1C[C@@H](n2cnc3c(Cl)nc(Cl)nc32)[C@@H](O)[C@@H]1O

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AHCY P23526 8/20 0.57
LMNA P02545 2/20 0.50
TP53 P04637 2/20 0.50
ADORA3 P0DMS8 5/20 0.48
ADORA2A P29274 2/20 0.48
ADORA1 P30542 2/20 0.48
PNP P00491 1/20 0.41
HTT P42858 1/20 0.41
PDE4D Q08499 1/20 0.41
PDE3A Q14432 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL293325 1.00 AHCY (0.57) AHCYLMNATP53ADORA3ADORA2A
SCHEMBL1841287 1.00 AHCY (0.57) AHCYLMNATP53ADORA3ADORA2A
SCHEMBL243600 1.00 AHCY (0.57) AHCYLMNATP53ADORA3ADORA2A
Trifluoroacetic Acid SCHEMBL1412146 0.90 AHCY (0.48) AHCYLMNATP53ADORA3ADORA2A
Trifluoroacetic Acid SCHEMBL241441 0.90 AHCY (0.48) AHCYLMNATP53ADORA3ADORA2A
SCHEMBL26381988 0.86 AHCY (0.57) AHCYLMNATP53ADORA3ADORA2A
SCHEMBL13211900 0.86 AHCY (0.54) AHCYADORA3ADORA2AADORA1
SCHEMBL12050237 0.84 AHCY (0.56) AHCYLMNATP53ADORA3ADORA2A
SCHEMBL8960194 0.84 AHCY (0.56) AHCYLMNATP53ADORA3ADORA2A
SCHEMBL3007619 0.83 LMNA (0.46) AHCYLMNATP53ADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2013211-B1 PURINE DERIVATIVES FOR USE AS ADENOSIN A2A RECEPTOR AGONISTS NOVARTIS AG (CH) 2012-03-14 EP disclosed