SCHEMBL2933263

SCHEMBL2933263

C[C@@H](c1ccc(-c2cc(OC(N)=O)c(NC(N)=O)s2)cc1)N1CCOCC1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 9/20 0.42
LRRK2 Q5S007 1/20 0.40
IKBKB O14920 3/20 0.38
JAK2 O60674 2/20 0.37
MEN1 O00255 1/20 0.37
EIF2AK2 P19525 1/20 0.37
KMT2A Q03164 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
MAPT P10636 1/20 0.37
MCL1 Q07820 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
ABCC1 P33527 1/20 0.36
JAK3 P52333 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2928533 1.00 CHEK1 (0.42) CHEK1LRRK2IKBKBJAK2MEN1
SCHEMBL2933488 0.90 CHEK1 (0.45) CHEK1IKBKBJAK2MEN1EIF2AK2
SCHEMBL1928818 0.85 IKBKB (0.55) CHEK1IKBKBJAK2MEN1EIF2AK2
SCHEMBL1928820 0.85 IKBKB (0.55) CHEK1IKBKBJAK2MEN1EIF2AK2
SCHEMBL1928275 0.85 IKBKB (0.55) CHEK1IKBKBJAK2MEN1EIF2AK2
SCHEMBL2927139 0.80 CHEK1 (0.41) CHEK1IKBKBJAK2MEN1EIF2AK2
SCHEMBL2934362 0.80 CHEK1 (0.58) CHEK1IKBKBJAK2MEN1KMT2A
SCHEMBL2931062 0.77 CHEK1 (0.59) CHEK1IKBKBJAK2JAK3
SCHEMBL2932975 0.77 PTGER1 (0.43) CHEK1JAK2MEN1KMT2AMAPT
SCHEMBL2933735 0.76 CHEK1 (0.44) CHEK1JAK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1421074-B1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2010-09-29 EP claimed