SCHEMBL29339728

SCHEMBL29339728

CC(C)(C)c1cc2cc(N)ccc2cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.41
HSD17B10 Q99714 4/20 0.41
CYP3A4 P08684 3/20 0.41
CASP1 P29466 3/20 0.41
HIF1A Q16665 3/20 0.41
TDP1 Q9NUW8 2/20 0.41
CASP7 P55210 2/20 0.41
HBB P68871 2/20 0.41
ALOX15 P16050 1/20 0.41
KDM4E B2RXH2 8/20 0.39
LMNA P02545 3/20 0.39
POLB P06746 2/20 0.39
CASP6 P55212 1/20 0.39
EGFR P00533 2/20 0.38
PLAU P00749 1/20 0.37
MEN1 O00255 5/20 0.36
KMT2A Q03164 5/20 0.36
HTT P42858 4/20 0.36
F2 P00734 1/20 0.36
CHRM2 P08172 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10220695 0.81 CYP1A2 (0.50) ALDH1A1HSD17B10TDP1KDM4ELMNA
SCHEMBL16937572 0.79 NR1I2 (0.37) ALDH1A1HSD17B10TDP1ALOX15LMNA
SCHEMBL10220696 0.78 GSK3A (0.42) ALDH1A1KDM4ELMNAMEN1KMT2A
SCHEMBL22244079 0.78 CCR9 (0.40) ALDH1A1TDP1KDM4EHTTMAPT
SCHEMBL27097160 0.78 CASP3 (0.46) TDP1MAPT
SCHEMBL762341 0.76 CYP1A2 (0.54) TDP1KDM4ELMNAPLAURAB9A
SCHEMBL14072410 0.75 UGT2B7 (0.34) ALDH1A1CYP3A4HIF1ALMNAMEN1
SCHEMBL25917123 0.75 RAB9A (0.50) CYP3A4EGFRRAB9ANPC1
SCHEMBL19089948 0.75
SCHEMBL25917114 0.75 CYP1A2 (0.44) ALDH1A1LMNAMEN1KMT2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240239752-A1 BICYCLIC HETEROAROMATIC INHIBITORS OF KLK5 WILMINGTON TRUST, NATIONAL ASSOCIATION 2024-07-18 US disclosed
US-20240239752-A1 BICYCLIC HETEROAROMATIC INHIBITORS OF KLK5 WILMINGTON TRUST, NATIONAL ASSOCIATION 2024-07-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240239752-A1 BICYCLIC HETEROAROMATIC INHIBITORS OF KLK5 KLK5, KLK1, KLKB1 ALDH1A1 1532/4885HSD17B10 169/4885CYP3A4 630/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.