SCHEMBL2934704

SCHEMBL2934704

CC(c1ccccc1)c1cccc(C(N)=O)c1C=O.c1ccc2c(c1)CO2

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 7/20 0.36
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ALOX12 P18054 1/20 0.35
AURKA O14965 2/20 0.32
RPS6KB1 P23443 2/20 0.32
AURKB Q96GD4 1/20 0.32
CYP11B1 P15538 2/20 0.32
CYP11B2 P19099 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5968855 0.72 IRAK4 (0.47) PARP1MAPTAURKARPS6KB1AURKB
SCHEMBL3663651 0.72 IRAK4 (0.47) PARP1MAPTAURKARPS6KB1AURKB
SCHEMBL6266294 0.72 IRAK4 (0.47) PARP1MAPTAURKARPS6KB1AURKB
SCHEMBL27511285 0.70 IRAK4 (0.42) PARP1MAPTAURKARPS6KB1AURKB
SCHEMBL21835618 0.70 IRAK4 (0.42) PARP1MAPTAURKARPS6KB1AURKB
SCHEMBL20425250 0.70 IRAK4 (0.42) PARP1MAPTAURKARPS6KB1AURKB
SCHEMBL4560229 0.68 BCAT2 (0.45) PARP1AURKARPS6KB1AURKB
SCHEMBL28754510 0.67 CTNNB1 (0.47) PARP1TP53MAPTSMN1; SMN2
SCHEMBL3351170 0.66 IRAK4 (0.47) PARP1MAPTAURKARPS6KB1AURKB
SCHEMBL4786305 0.66 IRAK4 (0.47) PARP1MAPTAURKARPS6KB1AURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1313731-B1 THIAZOLIDINE DERIVATIVES AND ITS USE AS ANTIFUNGAL AGENT UCB SA (BE) 2010-09-29 EP disclosed
EP-1313731-A1 THIAZOLIDINE DERIVATIVES AND ITS USE AS ANTIFUNGAL AGENT Oxford GlycoSciences (UK) Limited (GB) 2003-05-28 EP disclosed
WO-2002022612-A1 THIAZOLIDINE DERIVATIVES AND ITS USE AS ANTIFUNGAL AGENT OXFORD GLYCOSCIENCES (UK) LIMITED (GB) 2002-03-21 WO disclosed