SCHEMBL2934834

SCHEMBL2934834

O=C(O)CN1C(=O)C(Cc2ccccc2)NC12CCN(C(=O)c1ccc3ccccc3c1)CC2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.48
DRD4 P21917 3/20 0.47
ACHE P22303 1/20 0.45
TSHR P16473 2/20 0.43
LMNA P02545 2/20 0.43
RAB9A P51151 1/20 0.43
HPGD P15428 1/20 0.42
AKR1C1 Q04828 1/20 0.42
TPSAB1 Q15661 1/20 0.41
TPSD1 Q9BZJ3 1/20 0.41
TPSG1 Q9NRR2 1/20 0.41
CAPN1 P07384 1/20 0.40
CTSB P07858 1/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
USP2 O75604 1/20 0.39
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1807471 0.91 NPC1 (0.54) NPC1DRD4ACHETSHRLMNA
Hydrochloric Acid SCHEMBL1811368 0.91 NPC1 (0.53) NPC1DRD4ACHETSHRLMNA
SCHEMBL2942653 0.88 HPGD (0.42) TSHRLMNAHPGDALDH1A1GAA
SCHEMBL2941530 0.87 HPGD (0.43) TSHRLMNAHPGDALDH1A1NPSR1
SCHEMBL2940005 0.85 MGLL (0.43) TSHRHPGDALDH1A1GAAHTT
SCHEMBL2943001 0.84 MEN1 (0.39) TSHRGAA
SCHEMBL2940506 0.84 CYP3A4 (0.40) TSHRUSP2ALDH1A1GAA
SCHEMBL2942520 0.84 CYP3A4 (0.58) LMNAHPGDUSP2ALDH1A1GAA
SCHEMBL2940806 0.83 CA1 (0.56) CA12CA1CA2CA7CA9
SCHEMBL2942498 0.83 AVPR1A (0.53) LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730147-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO[4,5]DECAN-2-ON COMPOUNDS FOR USE IN THE TREATMENT OF OBESITY GRUENENTHAL GMBH (DE) 2010-02-03 EP claimed