Cediranib

Cediranib

SCHEMBL29351458

COc1cc2c(Oc3ccc4[nH]c(C)cc4c3F)ncnc2cc1OCCCN1CCCC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

FLT1FLT4KDRKITPDGFRAPDGFRB

The experimentally established mechanism targets of Cediranib. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR known ✓ P35968 11/20 1.00
FLT4 known ✓ P35916 5/20 1.00
FLT1 known ✓ P17948 4/20 1.00
PDGFRB known ✓ P09619 2/20 1.00
KIT known ✓ P10721 1/20 1.00
PDGFRA known ✓ P16234 1/20 1.00
RET P07949 4/20 1.00
TEK Q02763 2/20 1.00
AURKB Q96GD4 2/20 1.00
PLK4 O00444 1/20 1.00
GAK O14976 1/20 1.00
EPHB6 O15197 1/20 1.00
RIPK2 O43353 1/20 1.00
ERN1 O75460 1/20 1.00
STK10 O94804 1/20 1.00
MAP4K4 O95819 1/20 1.00
CHEK2 O96017 1/20 1.00
ABL1 P00519 1/20 1.00
EGFR P00533 1/20 1.00
ERBB2 P04626 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cediranib SCHEMBL63147 1.00 KDR (1.00) KDRFLT4RETFLT1PDGFRB
Cediranib SCHEMBL29368143 1.00 KDR (1.00) KDRFLT4RETFLT1PDGFRB
Cediranib SCHEMBL29383181 1.00 KDR (1.00) KDRFLT4RETFLT1PDGFRB
SCHEMBL1685423 0.99 ABCB11 (1.00) KDRFLT4RETFLT1PDGFRB
SCHEMBL20077514 0.94 KDR (0.89) KDRFLT4RETFLT1PDGFRB
Cediranib SCHEMBL4186434 0.94 KDR (0.89) KDRFLT4RETFLT1PDGFRB
SCHEMBL3198096 0.94 KDR (0.89) KDRFLT4RETFLT1PDGFRB
SCHEMBL13471998 0.94 KDR (0.89) KDRFLT4RETFLT1PDGFRB
SCHEMBL1401668 0.94 KDR (0.89) KDRFLT4RETFLT1PDGFRB
SCHEMBL1401641 0.93 KDR (0.88) KDRFLT4RETFLT1PDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 6884 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4071174-B1 METHODS COMPRISING FIXED INTERMITTENT DOSING OF CEDIRANIB ASTRAZENECA AB (SE) 2026-05-27 EP claimed
EP-4735045-A2 OXAZAPHOSPHORINE ANTIBODY DRUG CONJUGATES AND METHODS OF USE La Life Products, LLC (US) 2026-05-06 EP claimed
EP-4729519-A1 CRYSTAL FORM OF ENPP1 INHIBITOR CSPC Zhongqi Pharmaceutical Technology (Shijiazhuang) Co., Ltd. (CN) 2026-04-22 EP claimed
EP-4719387-A2 COMPLEMENT ANTIBODY-DRUG CONJUGATES ADS Therapeutics LLC (US) 2026-04-08 EP claimed
US-20260085061-A1 PHTHALAZINE DERIVATIVES AS PYRUVATE KINASE MODULATORS SITRYX THERAPEUTICS LIMITED (GB) 2026-03-26 US claimed
US-12576085-B2 Combination comprising an ATP analog and an adenosine receptor antagonist or a nucleobase/nucleoside analog for the treatment of cancer SAWYER MICHAEL BRUCE (CA) 2026-03-17 US claimed
US-12576077-B2 Composition for preventing, alleviating or treating cancer CKP THERAPEUTICS, INC. (US) 2026-03-17 US claimed
US-12577255-B2 MDM2-based modulators of proteolysis and associated methods of use ARVINAS OPERATIONS, INC. (US) 2026-03-17 US claimed
EP-4704832-A2 BIFUNCTIONAL SMALL MOLECULES TO TARGET THE SELECTIVE DEGRADATION OF CIRCULATING PROTEINS Biohaven Therapeutics Ltd. (VG) 2026-03-11 EP claimed
US-20260034056-A1 PHARMACEUTICAL COMPOSITIONS FOR TREATING OCULAR DISEASES OR DISORDERS ALCON INC (CH) 2026-02-05 US claimed
CN-114075159-A Purification method and application of olapari 吉林汇康制药有限公司 2022-02-22 CN claimed
WO-2022020720-A9 COMPOSITIONS AND METHODS FOR TREATING CANCER TCR2 Therapeutics Inc. (US) 2022-02-17 WO claimed
EP-3953390-A1 HUMAN ANTIBODIES THAT BIND RET AND METHODS OF USE THEREOF Regeneron Pharmaceuticals, Inc. (US) 2022-02-16 EP claimed
US-11246864-B2 Compositions and methods of using nintedanib for treating ocular diseases with abnormal neovascularization ADS THERAPEUTICS LLC (US) 2022-02-15 US claimed
WO-2022032113-A1 PHARMACEUTICALS FOR TREATING OR PREVENTING NIDOVIRUSES AND PICORNAVIRUSES THE UNIVERSITY OF CHICAGO (US) 2022-02-10 WO claimed
CN-114010787-A Compositions and methods for treating pterygium 拨云生物医药科技(广州)有限公司 2022-02-08 CN claimed
WO-2022026510-A1 METHODS OF TREATING HER2 POSITIVE CANCER WITH TUCATINIB IN COMBINATION WITH TRASTUZUMAB, A TAXANE, AND A VEGFR-2 ANTAGONIST SEAGEN INC. (US) 2022-02-03 WO claimed
CN-113993898-A Human antibodies that bind RET and methods of use thereof 瑞泽恩制药公司 2022-01-28 CN claimed
WO-2022020720-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER TCR2 Therapeutics Inc. (US) 2022-01-27 WO claimed
CN-113967261-A Application of FOLR1 inhibitor and medicine mixture for treating liver cancer 中国科学院大连化学物理研究所 2022-01-25 CN claimed