Sitravatinib

Sitravatinib

SCHEMBL29355690

COCCNCc1ccc(-c2cc3nccc(Oc4ccc(NC(=O)C5(C(=O)Nc6ccc(F)cc6)CC5)cc4F)c3s2)nc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 8/20 1.00
KDR P35968 8/20 1.00
AXL P30530 4/20 1.00
FLT3 P36888 2/20 1.00
NTRK1 P04629 1/20 1.00
KIT P10721 1/20 1.00
NTRK2 Q16620 1/20 1.00
MST1R Q04912 12/20 0.76
MERTK Q12866 2/20 0.76
PLK4 O00444 1/20 0.76
MAP4K4 O95819 1/20 0.76
ABL1 P00519 1/20 0.76
LCK P06239 1/20 0.76
FYN P06241 1/20 0.76
LYN P07948 1/20 0.76
HCK P08631 1/20 0.76
PDGFRB P09619 1/20 0.76
BCR P11274 1/20 0.76
SRC P12931 1/20 0.76
ABL2 P42684 1/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sitravatinib SCHEMBL29774217 1.00 MET (1.00) METKDRAXLFLT3NTRK1
Sitravatinib SCHEMBL172015 1.00 MET (1.00) METKDRAXLFLT3NTRK1
Sitravatinib SCHEMBL30276257 1.00 MET (1.00) METKDRAXLFLT3NTRK1
SCHEMBL23118344 0.96 MET (0.92) METKDRAXLFLT3NTRK1
SCHEMBL12557940 0.96 MET (0.92) METKDRAXLFLT3NTRK1
Sitravatinib SCHEMBL26109867 0.96 MET (0.91) METKDRAXLFLT3NTRK1
Sitravatinib SCHEMBL29927268 0.96 MET (0.91) METKDRAXLFLT3NTRK1
Sitravatinib SCHEMBL29910958 0.96 MET (0.91) METKDRAXLFLT3NTRK1
SCHEMBL2605829 0.95 MET (0.91) METKDRAXLFLT3NTRK1
SCHEMBL14817556 0.95 MET (0.91) METKDRAXLFLT3NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1021 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12559800-B2 KMT2A-MAML2 fusion molecules and uses thereof FOUNDATION MEDICINE, INC. (US) 2026-02-24 US claimed
EP-4694930-A1 COMBINATION THERAPIES INVOLVING GREM1 ANTAGONISTS FOR TREATMENT OF CANCER Suzhou Transcenta Therapeutics Co., Ltd. (CN) 2026-02-18 EP claimed
US-20250381202-A1 PRODRUG KIT FOR MULTI-PRONGED CHEMOTHERAPY ZOUNEK ALEX (DE) 2025-12-18 US claimed
EP-4653019-A1 ANTI-HER2 ANTIBODY-DRUG CONJUGATE FOR TREATING BREAST CANCER Jiangsu Hengrui Pharmaceuticals Co., Ltd. (CN) 2025-11-26 EP claimed
EP-3957329-B1 COMPOSITION COMPRISING THE COMBINATION OF SOTAGLIFLOZIN AS THE SODIUM/GLUCOSE CO-TRANSPORTER 1 INHIBITOR (SGLT1) AND A VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2 INHIBITOR (VEGFR2) FOR USE IN TREATING CANCER NEWISH TECH BEIJING CO LTD (CN) 2025-11-19 EP claimed
EP-4640714-A2 METHODS FOR ASSESSING RISK OF DEVELOPING A VIRAL DISEASE USING A GENETIC TEST PML Screening, LLC (US) 2025-10-29 EP claimed
EP-4637821-A1 HER3 RADIOIMMUNOTHERAPY FOR THE TREATMENT OF SOLID CANCERS Actinium Pharmaceuticals, Inc. (US) 2025-10-29 EP claimed
EP-4615506-A1 USE OF GSK-3 ACTIVATIOR TO MODULATE PROTEASOME ACTIVITY TO PREVENT AGEING ASSOCIATED CONDITIONS AND DISEASES Sahin, Fikret (TR) 2025-09-17 EP claimed
EP-3957631-B1 QUINOLINE COMPOUND OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF FOR TREATING EWING'S SARCOMA CHIA TAI TIANQING PHARMACEUTICAL GROUP CO LTD (CN) 2025-09-10 EP claimed
EP-4604920-A1 LYOPHILIZED FORMULATIONS OF CD73 COMPOUNDS Arcus Biosciences, Inc. (US) 2025-08-27 EP claimed
EP-3973963-A1 QUINOLINE DERIVATIVES FOR TREATMENT OF HEAD AND NECK CANCER Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2022-03-30 EP claimed
US-11285154-B2 Methods and compositions for treating cancer UNITED STATES GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS (US) 2022-03-29 US claimed
WO-2022060831-A1 COMBINATION THERAPIES Mirati Therapeutics, Inc. (US) 2022-03-24 WO claimed
EP-3967310-A1 QUINOLINE DERIVATIVE USED FOR SOFT TISSUE SARCOMA COMBINATION THERAPY CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD. (CN) 2022-03-16 EP claimed
EP-3964217-A1 USE OF COMPOUND OR PHARMACEUTICALLY ACCEPTABLE SALT, DIMER OR TRIMER THEREOF IN PREPARATION OF DRUG FOR TREATING CANCER Newish Technology (Beijing) Co., Ltd. (CN) 2022-03-09 EP claimed
WO-2022043816-A2 RATIONAL IDENTIFICATION OF FDA APPROVED DRUGS BY COMPUTATIONAL MODELLING AND INHIBITION OF RBD/ACE2 BINDING FOR TREATMENT OF COVID-19 REAGENE INNOVATIONS PVT. LTD. (IN) 2022-03-03 WO claimed
EP-3957310-A1 COMPOSITION AND USE THEREOF IN PREPARATION OF MEDICATION FOR TREATING CANCER Newish Technology (Beijing) Co., Ltd. (CN) 2022-02-23 EP claimed
EP-3957631-A1 QUINOLINE COMPOUND OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF FOR TREATING EWING'S SARCOMA Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2022-02-23 EP claimed
EP-3957329-A1 COMPOSITION FOR TREATING CANCER, APPLICATION THEREOF, AND DRUG Newish Technology (Beijing) Co., Ltd. (CN) 2022-02-23 EP claimed
EP-3942045-A1 A DBAIT MOLECULE IN COMBINATION WITH KINASE INHIBITOR FOR THE TREATMENT OF CANCER ONXEO (FR) 2022-01-26 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12559800-B2 KMT2A-MAML2 fusion molecules and uses thereof DNER, EGFR, NOTCH2 MET 9/4885KDR 498/4885AXL 727/4885
US-20250381202-A1 PRODRUG KIT FOR MULTI-PRONGED CHEMOTHERAPY KIT, CTSL, PAICS MET 124/4885KDR 328/4885AXL 497/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.