Aviptadil

Aviptadil

SCHEMBL29357337

CC[C@H](C)[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](CCSC)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(=O)O)NC(=O)[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@@H](N)Cc1cnc[nH]1)C(C)C)[C@@H](C)O)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(N)=O)C(=O)O

nearest known ligand 0.84

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2C

The experimentally established mechanism targets of Aviptadil. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
VIPR1 P32241 9/20 0.84
VIPR2 P41587 10/20 0.81
GLP1R P43220 5/20 0.73
CCKBR P32239 1/20 0.73
ECE1 P42892 1/20 0.69
MUS81 Q96NY9 1/20 0.69
PTH1R Q03431 2/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29382043 0.95 GLP1R (0.80) VIPR1VIPR2GLP1RCCKBRECE1
SCHEMBL29382033 0.94 GLP1R (0.78) VIPR1VIPR2GLP1RCCKBRECE1
Vasoactive Intestinal Peptide SCHEMBL30752406 0.93 VIPR1 (0.73) VIPR1VIPR2GLP1RCCKBRECE1
Vasoactive Intestinal Peptide SCHEMBL3041046 0.92 VIPR1 (0.72) VIPR1VIPR2GLP1RCCKBR
Aviptadil SCHEMBL30969141 0.92 VIPR1 (0.72) VIPR1VIPR2GLP1RCCKBR
SCHEMBL29496440 0.92 VIPR1 (0.71) VIPR1VIPR2GLP1RCCKBRPTH1R
Oxyntomodulin SCHEMBL29349603 0.92 GLP1R (0.84) VIPR1GLP1RCCKBRECE1MUS81
SCHEMBL30542042 0.91 VIPR1 (0.70) VIPR1VIPR2GLP1RCCKBRECE1
Spinigerin SCHEMBL29593748 0.91 VIPR2 (0.70) VIPR1VIPR2GLP1RCCKBRECE1
SCHEMBL29403715 0.90 VIPR1 (0.72) VIPR1VIPR2GLP1RCCKBRECE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 702 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4228644-B1 N-[4-[1-(1,4-DIOXASPIRO[4.5]DEC-8-YL)-4-(8-OXA-3-AZABICYCLO[3.2.1]OCT-3-YL)-1H-PYRAZOLO[3,4-D]PYRIMIDIN-6-YL]PHENYL]-N'-METHYLUREA FOR USE IN THE TREATMENT OF COVID19 NANTCELL INC (US) 2026-05-27 EP claimed
US-20260124148-A1 POLYPEPTIDE FORMULATIONS FOR ORAL DELIVERY BHAMIS RES LABORATORY PVT LTD (IN) 2026-05-07 US claimed
EP-4731243-A2 IN SITU THERAPEUTIC PRODUCTION: METHODS AND COMPOSITIONS William Marsh Rice University (US) 2026-04-29 EP claimed
EP-4725496-A2 N-[4-[1-(1,4-DIOXASPIRO[4.5]DEC-8-YL)-4-(8-OXA-3-AZABICYCLO[3.2.1]OCT-3-YL)-1H-PYRAZOLO[3,4-D]PYRIMIDIN-6-YL]PHENYL]-N'-METHYLUREA FOR USE IN THE TREATMENT OF COVID19 NantCell, Inc. (US) 2026-04-15 EP claimed
US-20260027062-A1 IMPROVED ORAL PHARMACEUTICAL FORMULATIONS OF THERAPEUTIC PEPTIDES AND PROTEINS CYPRUMED GMBH (AT) 2026-01-29 US claimed
US-12533321-B2 Polypeptide formulations for oral delivery Bhami's Research Laboratory, Pvt. Ltd. (IN) 2026-01-27 US claimed
US-12465605-B2 Methods and materials for gender-dependent treatment of cardiovascular dysfunction MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH (US) 2025-11-11 US claimed
WO-2025227105-A1 CLEAVABLE LINKERS WITH TUNABLE HALF-LIVES UNIVERSITY OF UTAH RESEARCH FOUNDATION (US) 2025-10-30 WO claimed
EP-4611721-A1 STABLE AVIPTADIL FORMULATIONS Relief Therapeutics International SA (CH) 2025-09-10 EP claimed
EP-4601623-A1 POLYPEPTIDE FORMULATIONS FOR ORAL DELIVERY Bhami's Research Laboratory, Pvt. Ltd. (IN) 2025-08-20 EP claimed
US-20220323546-A1 RECOMBINANT INTERFERON ALTUM PHARMACEUTICALS INC. (CA) 2022-10-13 US claimed
CN-115066254-A Human anti-inflammatory peptides for inhalation treatment of inflammatory lung diseases 阿德维塔生命科学有限责任公司 2022-09-16 CN claimed
US-20220175889-A1 NEW DOSAGE REGIMEN FOR INHALED VASOACTIVE INTESTINAL POLYPEPTIDE CENTURION ILAÇ SANAYI VE TICARET ANONIM SIRKETI (TR) 2022-06-09 US claimed
WO-2022119535-A1 NEW DOSAGE REGIMEN FOR INHALED VASOACTIVE INTESTINAL POLYPEPTIDE CENTURION ILAC SANAYI VE TICARET ANONIM SIRKETI (TR) 2022-06-09 WO claimed
WO-2022106984-A2 SMALL MOLECULE INHIBITORS OF SARS-COV2 MAIN PROTEASE NANTCELL, INC. (US) 2022-05-27 WO claimed
US-20220133630-A1 PREPARATION METHOD OF SUSTAINED-RELEASE MICROPARTICLES AC PHARMACEUTICALS CO., LTD. (CN) 2022-05-05 US claimed
WO-2022083853-A1 AGONISTS OF FREE FATTY ACID RECEPTOR 1 AND THEIR USE IN DISEASES ASSOCIATED WITH SAID RECEPTOR GBIOTECH S.À.R.L. (CH) 2022-04-28 WO claimed
WO-2022081406-A1 PHARMACEUTICALS FOR COVID19 TREATMENT IMMUNITYBIO, INC. (US) 2022-04-21 WO claimed
WO-2022076903-A1 NIRAN INTERFERING DRUGS FOR SARS-COV-2 MUTANT THERAPY Atea Pharmaceuticals, Inc. (US) 2022-04-14 WO claimed
WO-2022028917-A2 METHODS FOR THE DETERMINATION OF THE PREDISPOSITION FOR A SEVERE OR CRITICAL COURSE OF A COVID-19-DISEASE FROM A MILD OR MODERATE COURSE OF A COVID-19-DISEASE IN A SUBJECT SCIOMICS GMBH (DE) 2022-02-10 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12533321-B2 Polypeptide formulations for oral delivery PTMS, IAPP, IGF1R VIPR1 3306/4885VIPR2 2742/4885GLP1R 4/4885
US-20260027062-A1 IMPROVED ORAL PHARMACEUTICAL FORMULATIONS OF THERAPEUTIC PEPTIDES AND PROTEINS ADM2, TAS2R42, ACP1 VIPR1 874/4885VIPR2 685/4885GLP1R 130/4885
US-20260124148-A1 POLYPEPTIDE FORMULATIONS FOR ORAL DELIVERY GLP1R, TTR, IAPP VIPR1 813/4885VIPR2 565/4885GLP1R 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.