SCHEMBL29360805

SCHEMBL29360805

Cc1cc2ncccc2c(F)c1Br

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.41
MAPT P10636 1/20 0.41
ATAD2 Q6PL18 1/20 0.39
CCR1 P32246 1/20 0.39
CCR8 P51685 1/20 0.39
CYP1A2 P05177 2/20 0.38
CYP1B1 Q16678 1/20 0.38
NR4A2 P43354 1/20 0.38
NPC1 O15118 2/20 0.37
HSP90AA1 P07900 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HTT P42858 3/20 0.37
ALDH1A1 P00352 2/20 0.37
CYP2C19 P33261 1/20 0.37
SYK P43405 1/20 0.36
BRD4 O60885 1/20 0.36
NSD2 O96028 1/20 0.36
CASP6 P55212 1/20 0.36
PSMD14 O00487 1/20 0.35
COPS5 Q92905 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28724330 1.00 KDM4E (0.41) KDM4EMAPTATAD2CCR1CCR8
SCHEMBL1161526 0.82 KDM4E (0.43) KDM4EMAPTCYP1A2NR4A2NPC1
SCHEMBL11985966 0.79 NPC1 (0.44) KDM4EMAPTATAD2CCR1CCR8
SCHEMBL14205600 0.77 MET (0.41) KDM4EMAPTATAD2CCR1CCR8
SCHEMBL13676646 0.77 KDM4E (0.38) KDM4EMAPTATAD2CCR1CCR8
SCHEMBL13676597 0.77 KDM4E (0.38) KDM4EMAPTATAD2CCR1CCR8
SCHEMBL29363534 0.76 L3MBTL1 (0.41) KDM4EMAPTCCR1CCR8CYP1A2
SCHEMBL243422 0.76 HTT (0.45) KDM4EMAPTATAD2CCR1CCR8
SCHEMBL28724331 0.76 L3MBTL1 (0.41) KDM4EMAPTCCR1CCR8CYP1A2
SCHEMBL12121755 0.75 L3MBTL1 (0.44) KDM4EMAPTCCR1CCR8CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022017368-A1 DNA-PK SELECTIVE INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF 首药控股(北京)股份有限公司 2022-01-27 WO disclosed