Bfh-772

Bfh-772

SCHEMBL29366190

O=C(Nc1cccc(C(F)(F)F)c1)c1cccc2cc(Oc3cc(CO)ncn3)ccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

KDR

The experimentally established mechanism targets of Bfh-772. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDR known ✓ P35968 19/20 1.00
FLT1 P17948 5/20 1.00
FLT4 P35916 5/20 1.00
RET P07949 2/20 1.00
PDGFRB P09619 2/20 1.00
KIT P10721 2/20 1.00
RXFP1 Q9HBX9 1/20 0.51
MAPK14 Q16539 3/20 0.51
TNNI3K Q59H18 3/20 0.51
BRAF P15056 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bfh-772 SCHEMBL987715 1.00 KDR (1.00) KDRFLT1FLT4RETPDGFRB
Bfh-772 SCHEMBL1041162 0.99 KDR (0.98) KDRFLT1FLT4RETPDGFRB
SCHEMBL2465073 0.93 KDR (0.87) KDRFLT1FLT4RETPDGFRB
SCHEMBL2435271 0.92 KDR (0.85) KDRFLT1FLT4RETPDGFRB
SCHEMBL2434211 0.92 KDR (0.85) KDRFLT1FLT4RETPDGFRB
SCHEMBL2439589 0.91 KDR (0.83) KDRFLT1FLT4RETPDGFRB
SCHEMBL2468872 0.91 KDR (0.83) KDRFLT1FLT4RETPDGFRB
SCHEMBL2438656 0.90 KDR (0.81) KDRFLT1FLT4RETPDGFRB
SCHEMBL2437180 0.90 KDR (0.81) KDRFLT1FLT4RETPDGFRB
SCHEMBL1875161 0.89 KDR (0.80) KDRFLT1FLT4RETPDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 94 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4539924-A1 COMPOSITIONS, SYSTEMS, AND METHODS FOR TREATING CANCER USING TUMOR TREATING FIELDS AND VEGF INHIBITORS Novocure GmbH (CH) 2025-04-23 EP claimed
CN-119451723-A Compositions, systems, and methods for treating cancer using a tumor treating electric field and a VEGF inhibitor 诺沃库勒有限责任公司 2025-02-14 CN claimed
WO-2023248139-A1 COMPOSITIONS, SYSTEMS, AND METHODS FOR TREATING CANCER USING TUMOR TREATING FIELDS AND VEGF INHIBITORS NOVOCURE GMBH (CH) 2023-12-28 WO claimed
US-20230405316-A1 COMPOSITIONS, SYSTEMS, AND METHODS FOR TREATING CANCER USING TUMOR TREATING FIELDS AND VEGF INHIBITORS NOVOCURE GMBH (CH) 2023-12-21 US claimed
CN-114585356-A Methods of preventing or treating diseases associated with VEGFR and/or VEGF inhibition 上海岸阔医药科技有限公司 2022-06-03 CN claimed
CN-114028568-A Method for preventing or treating side effects of tumor therapy 上海岸阔医药科技有限公司 2022-02-11 CN claimed
CN-113975264-A Method for preventing or treating side effects of tumor therapy 上海岸阔医药科技有限公司 2022-01-28 CN claimed
CN-122094689-A Combination therapy of diacylglycerol kinase (DGK) alpha inhibitors with other therapies 2026-05-26 CN disclosed
EP-4739310-A1 ECTONUCLEOTIDE PYROPHOSPHATASE/PHOSPHODIESTERASE 1 (ENPP1) INHIBITOR COMBINATIONS AND USES THEREOF Insilico Medicine IP Limited (HK) 2026-05-13 EP disclosed
US-12599664-B2 Pharmaceutical products and stable liquid compositions of IL-17 antibodies NOVARTIS AG (CH) 2026-04-14 US disclosed
US-12594331-B2 Methods of treating psoriasis with secukinumab NOVARTIS AG (CH) 2026-04-07 US disclosed
US-12594332-B2 Methods of treating psoriasis with secukinumab NOVARTIS AG (CH) 2026-04-07 US disclosed
US-20260083842-A1 PHARMACEUTICAL PRODUCTS AND STABLE LIQUID COMPOSITIONS OF IL-17 ANTIBODIES NOVARTIS AG (CH) 2026-03-26 US disclosed
US-11351253-B2 Methods of treating palmoplantar pustular psoriasis (PPP) using IL-17 antibody NOVARTIS AG (CH) 2022-06-07 US disclosed
CN-114585356-A Methods of preventing or treating diseases associated with VEGFR and/or VEGF inhibition 上海岸阔医药科技有限公司 2022-06-03 CN disclosed
EP-4003508-A1 PERFUSION MODULATED TUMOR DOSE SCULPTING WITH SINGLE DOSE RADIOTHERAPY Memorial Sloan Kettering Cancer Center (US) 2022-06-01 EP disclosed
CN-114452381-A Pharmaceutical product and stable liquid composition of IL-17 antibody 诺华股份有限公司 2022-05-10 CN disclosed
CN-114452380-A Pharmaceutical product and stable liquid composition of IL-17 antibody 诺华股份有限公司 2022-05-10 CN disclosed
CN-114028568-A Method for preventing or treating side effects of tumor therapy 上海岸阔医药科技有限公司 2022-02-11 CN disclosed
CN-113975264-A Method for preventing or treating side effects of tumor therapy 上海岸阔医药科技有限公司 2022-01-28 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260083842-A1 PHARMACEUTICAL PRODUCTS AND STABLE LIQUID COMPOSITIONS OF IL-17 ANTIBODIES IL17A, RAB7A, IL15 KDR 2616/4885FLT1 2741/4885FLT4 1709/4885
US-12599664-B2 Pharmaceutical products and stable liquid compositions of IL-17 antibodies IL17A, IL15, IL5 KDR 1367/4885FLT1 856/4885FLT4 598/4885
US-12594332-B2 Methods of treating psoriasis with secukinumab IL17A, IL15, IL23R KDR 535/4885FLT1 50/4885FLT4 86/4885
US-12594331-B2 Methods of treating psoriasis with secukinumab IL17A, IL15, IL15RA KDR 1107/4885FLT1 81/4885FLT4 136/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.