SCHEMBL29366337

SCHEMBL29366337

Cc1csc(-c2nc(-n3ncc4cnccc43)c3nc[nH]c3n2)n1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 5/20 0.35
TGFBR2 P37173 3/20 0.35
CYP2E1 P05181 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2A6 P11509 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2B6 P20813 1/20 0.34
PDE10A Q9Y233 2/20 0.34
TSHR P16473 1/20 0.33
MKNK2 Q9HBH9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23007811 1.00 TGFBR1 (0.35) TGFBR1TGFBR2CYP2E1CYP3A4CYP2A6
SCHEMBL23007807 0.82 TGFBR1 (0.43) TGFBR1TGFBR2CYP2A6PDE10A
SCHEMBL29366477 0.82 TGFBR1 (0.43) TGFBR1TGFBR2CYP2A6PDE10A
SCHEMBL29363247 0.75 TGFBR1 (0.35) TGFBR1PDE10AMKNK2
SCHEMBL23007890 0.75 TGFBR1 (0.35) TGFBR1PDE10AMKNK2
SCHEMBL23007722 0.73 TGFBR1 (0.39) TGFBR1TGFBR2CYP3A4MKNK2
SCHEMBL29366031 0.73 TGFBR1 (0.39) TGFBR1TGFBR2CYP3A4MKNK2
SCHEMBL23007810 0.72 CNR2 (0.39) TGFBR1
SCHEMBL29365713 0.72 CNR2 (0.39) TGFBR1
SCHEMBL23007796 0.67 TGFBR1 (0.36) TGFBR1TGFBR2MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113993870-B Imidazo pyrimidine compound containing fused ring group, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2023-06-13 CN disclosed
CN-113993870-A Imidazo pyrimidine compound containing polycyclic group, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2022-01-28 CN disclosed