SCHEMBL29367113

SCHEMBL29367113

COC[C@H](NC(=O)c1ccccc1)c1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.67
TAS1R1 Q7RTX1 1/20 0.67
NAMPT P43490 1/20 0.62
TACR3 P29371 1/20 0.55
ROCK2 O75116 4/20 0.55
ROCK1 Q13464 3/20 0.55
KDM4E B2RXH2 1/20 0.54
GAA P10253 1/20 0.54
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
UTS2R Q9UKP6 1/20 0.50
MAPK13 O15264 1/20 0.49
RPS6KA5 O75582 1/20 0.49
MAP4K4 O95819 1/20 0.49
PAK4 O96013 1/20 0.49
PRKCG P05129 1/20 0.49
CDK1 P06493 1/20 0.49
PRKACA P17612 1/20 0.49
RPS6KB1 P23443 1/20 0.49
CDK2 P24941 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3101155 0.85 ROCK2 (0.73) TAS1R3TAS1R1NAMPTROCK2ROCK1
SCHEMBL4490832 0.85 TAS1R3 (0.60) TAS1R3TAS1R1NAMPTTACR3ROCK2
SCHEMBL7723793 0.83 TAS1R3 (0.56) TAS1R3TAS1R1NAMPTTACR3ROCK2
SCHEMBL7723790 0.83 TAS1R3 (0.56) TAS1R3TAS1R1NAMPTTACR3ROCK2
SCHEMBL792022 0.83 TAS1R3 (0.56) TAS1R3TAS1R1NAMPTTACR3ROCK2
SCHEMBL1139148 0.83 MEN1 (0.53) TAS1R3TAS1R1NAMPTTACR3ROCK2
SCHEMBL14198862 0.83 MEN1 (0.63) TAS1R3TAS1R1TACR3ROCK2ROCK1
SCHEMBL12226572 0.83 MEN1 (0.63) TAS1R3TAS1R1TACR3ROCK2ROCK1
SCHEMBL27781112 0.83 MEN1 (0.63) TAS1R3TAS1R1TACR3ROCK2ROCK1
SCHEMBL15716619 0.82 TAS1R3 (0.54) TAS1R3TAS1R1NAMPTTACR3ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109983016-B Pyrimido [5,4-b ] indolizine or pyrimido [5,4-b ] pyridine compound, preparation method and application thereof 中国科学院上海药物研究所 2022-02-01 CN disclosed