SCHEMBL29368486

SCHEMBL29368486

COc1ccc(-c2nc(N)nc3ccccc23)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 8/20 1.00
NUDT1 P36639 3/20 0.70
SCN9A Q15858 1/20 0.68
LMNA P02545 2/20 0.61
KDM4E B2RXH2 1/20 0.61
ALDH1A1 P00352 1/20 0.61
NPSR1 Q6W5P4 1/20 0.61
TDP1 Q9NUW8 1/20 0.61
L3MBTL1 Q9Y468 1/20 0.61
ADORA1 P30542 2/20 0.61
CYP1A1 P04798 1/20 0.58
CYP1A2 P05177 1/20 0.58
CYP1B1 Q16678 1/20 0.58
MAPT P10636 1/20 0.58
MAPK1 P28482 1/20 0.58
APP P05067 1/20 0.56
ADORA3 P0DMS8 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12281655 0.83 ADORA2A (0.92) ADORA2ANUDT1SCN9AADORA1MAPT
SCHEMBL421987 0.83 ADORA2A (1.00) ADORA2ANUDT1SCN9AALDH1A1CYP1A2
SCHEMBL28872938 0.83 ADORA2A (0.70) ADORA2ALMNAKDM4EALDH1A1NPSR1
SCHEMBL15561039 0.82 LMNA (0.72) ADORA2ALMNAKDM4EALDH1A1NPSR1
Hydrochloric Acid SCHEMBL27344186 0.81 ADORA2A (0.96) ADORA2ANUDT1SCN9AALDH1A1CYP1A2
SCHEMBL28147437 0.81 ADORA2A (0.68) ADORA2ALMNAKDM4EALDH1A1NPSR1
SCHEMBL1289729 0.81 SCN9A (1.00) ADORA2ANUDT1SCN9A
SCHEMBL6768236 0.78 ADORA2A (0.63) ADORA2ANUDT1SCN9AKDM4EALDH1A1
SCHEMBL6695603 0.77 RAD52 (0.74) ADORA2ASCN9ALMNAKDM4EALDH1A1
SCHEMBL4108639 0.77 ADORA2A (0.63) ADORA2ANUDT1LMNAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113999180-A Quinazoline compound, intermediate thereof, preparation method, pharmaceutical composition and application 上海医药集团股份有限公司 2022-02-01 CN disclosed