SCHEMBL6768236

SCHEMBL6768236

COc1ccc2c(-c3ccc(S(=O)(=O)c4ccccc4)cc3)nc(N)nc2c1

nearest known ligand 0.63

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 10/20 0.63
SCN9A Q15858 1/20 0.47
NUDT1 P36639 1/20 0.46
ADORA1 P30542 4/20 0.45
DHFR P00374 2/20 0.45
MAPT P10636 2/20 0.44
TP53 P04637 1/20 0.44
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ADORA2B P29275 1/20 0.43
CASR P41180 1/20 0.42
FFAR2 O15552 1/20 0.41
ACACA Q13085 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30979864 0.79 ADORA2A (0.74) ADORA2ASCN9ANUDT1ADORA1DHFR
SCHEMBL29368486 0.78 ADORA2A (1.00) ADORA2ASCN9ANUDT1ADORA1MAPT
SCHEMBL8368164 0.76 ADORA2A (0.47) ADORA2ASCN9ANUDT1DHFRMAPT
SCHEMBL1884625 0.73 ADORA2A (0.64) ADORA2ANUDT1ADORA1DHFRMAPT
SCHEMBL29371576 0.73 ADORA2A (0.66) ADORA2ASCN9ANUDT1DHFR
SCHEMBL5619409 0.72 PDE4B (0.48) ADORA2ADHFR
SCHEMBL6027816 0.71 ADORA2A (0.62) ADORA2ASCN9ANUDT1ADORA1DHFR
SCHEMBL2900381 0.70 PKM (0.83) ALDH1A1SMN1; SMN2
SCHEMBL5384654 0.70 ALDH1A1 (0.64) MAPTTP53ALDH1A1KDM4ESMN1; SMN2
SCHEMBL14820340 0.69 DHFR (0.69) ADORA1DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6727256-B1 4-AMINOQUINAZOLINE DERIVATIVES AS ANTICARCINOGENIC AGENTS SMITHKLINE BEECHAM CORPORATION 2004-04-27 US disclosed