Bisindolylmaleimide Ix

Bisindolylmaleimide Ix

SCHEMBL29370657

Cn1cc(C2=C(c3cn(CCCSC(=N)N)c4ccccc34)C(=O)NC2=O)c2ccccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 4/20 1.00
PRKCB P05771 3/20 1.00
PRKCE Q02156 3/20 1.00
PIM1 P11309 3/20 1.00
MEN1 O00255 2/20 1.00
TP53 P04637 2/20 1.00
CYP3A4 P08684 2/20 1.00
MAPT P10636 2/20 1.00
ALOX15 P16050 2/20 1.00
TSHR P16473 2/20 1.00
MAPK1 P28482 2/20 1.00
RECQL P46063 2/20 1.00
KMT2A Q03164 2/20 1.00
SMN1; SMN2 Q16637 2/20 1.00
HIPK1 Q86Z02 2/20 1.00
SIRT2 Q8IXJ6 2/20 1.00
SIRT1 Q96EB6 2/20 1.00
HSD17B10 Q99714 2/20 1.00
SIRT3 Q9NTG7 2/20 1.00
TDP1 Q9NUW8 2/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bisindolylmaleimide Ix SCHEMBL1567017 1.00 PRKCA (1.00) PRKCAPRKCBPRKCEPIM1MEN1
Bisindolylmaleimide Ix SCHEMBL29381390 0.95 MEN1 (1.00) PRKCAPRKCBPRKCEPIM1MEN1
Bisindolylmaleimide Ix SCHEMBL2491726 0.95 MEN1 (1.00) PRKCAPRKCBPRKCEPIM1MEN1
SCHEMBL8166772 0.93 MEN1 (0.95) PRKCAPRKCBPRKCEPIM1MEN1
SCHEMBL8161675 0.92 MEN1 (0.93) PRKCAPRKCBPRKCEPIM1MEN1
SCHEMBL15600252 0.91 PIM1 (0.83) PRKCAPRKCBPRKCEPIM1MEN1
SCHEMBL18134615 0.90 PIM1 (0.81) PRKCAPRKCBPRKCEPIM1MEN1
SCHEMBL8154377 0.89 MEN1 (0.89) PRKCAPRKCBPRKCEPIM1MEN1
SCHEMBL8160916 0.88 PIM1 (0.78) PRKCAPRKCBPRKCEPIM1MEN1
SCHEMBL9088345 0.86 PRKCB (0.76) PRKCAPRKCBPRKCEPIM1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 362 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4627062-A1 CULTURE MEDIUM, COATING MATRIX AND METHOD FOR EXPANDING MIDBRAIN DOPAMINERGIC PROGENITOR CELLS Nuwacell Biotechnologies Co., Ltd. (CN) 2025-10-08 EP claimed
WO-2025120106-A1 METHODS FOR ISOLATING EMBRYONIC STEM CELLS FROM AN AVIAN EMBRYO CELLS SUPRÊME (FR) 2025-06-12 WO claimed
EP-4567102-A1 METHODS FOR ISOLATING EMBRYONIC STEM CELLS FROM AVIAN EMBRYONIC CELLS Suprême (FR) 2025-06-11 EP claimed
US-20250163388-A1 METHODS FOR DERIVATION AND PROPAGATION OF AVIAN PLURIPOTENT STEM CELLS AND APPLICATIONS THEREOF UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2025-05-22 US claimed
US-12215355-B2 Stem cell derived islet differentiation VERTEX PHARMACEUTICALS INCORPORATED (US) 2025-02-04 US claimed
US-12188046-B2 Culture medium, coating matrix and method for expanding midbrain dopaminergic progenitor cells NUWACELL BIOTECHNOLOGIES CO., LTD. (CN) 2025-01-07 US claimed
EP-4479521-A2 METHODS FOR DERIVATION AND PROPAGATION OF AVIAN PLURIPOTENT STEM CELLS AND APPLICATIONS THEREOF University of Southern California (US) 2024-12-25 EP claimed
EP-4461806-A2 SC-B CELLS AND COMPOSITIONS AND METHODS FOR GENERATING THE SAME President and Fellows of Harvard College (US) 2024-11-13 EP claimed
US-20240358767-A1 STEM CELL DIFFERENTIATION AND CHEMICAL COMPOUNDS VERTEX PHARMACEUTICALS INCORPORATED (US) 2024-10-31 US claimed
US-20240352413-A1 ISOLATED HUMAN LUNG PROGENITOR CELLS AND USES THEREOF THE GENERAL HOSPITAL CORPORATION (US) 2024-10-24 US claimed
US-20230201173-A1 SMAD4 Complex Inducers and Uses in Cancer Therapy UNIV EMORY (US) 2023-06-29 US claimed
WO-2023081884-A2 STEM CELL DIFFERENTIATION AND CHEMICAL COMPOUNDS VERTEX PHARMACEUTICALS INCORPORATED (US) 2023-05-11 WO claimed
US-20230079757-A1 METHODS AND MATERIALS FOR TREATING CANCER MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH 2023-03-16 US claimed
US-20230031009-A1 TREATMENT FOR CHEMOBRAIN UNIV YALE (US) 2023-02-02 US claimed
EP-4107278-A1 METHODS AND MATERIALS FOR TREATING CANCER Mayo Foundation for Medical Education and Research (US) 2022-12-28 EP claimed
US-20220378782-A1 KCC2 EXPRESSION ENHANCING COMPOUNDS AND USES THEREOF WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2022-12-01 US claimed
WO-2022192300-A1 STEM CELL DIFFERENTIATION AND POLYMERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-09-15 WO claimed
WO-2022147056-A1 ENHANCED DIFFERENTIATION OF BETA CELLS VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-07-07 WO claimed
WO-2022120187-A2 METHOD OF DETERMINING RESISTANCE TO CHECKPOINT INHIBITOR THERAPIES SHATTUCK LABS, INC. (US) 2022-06-09 WO claimed
US-20220162562-A1 SC-BETA CELLS AND COMPOSITIONS AND METHODS FOR GENERATING THE SAME HARVARD COLLEGE (US) 2022-05-26 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220378782-A1 KCC2 EXPRESSION ENHANCING COMPOUNDS AND USES THEREOF MECP2, SLC1A2, GRIN2C PRKCA 430/4885PRKCB 296/4885PRKCE 432/4885
US-20240358767-A1 STEM CELL DIFFERENTIATION AND CHEMICAL COMPOUNDS EBP, AKT3, PRKCD PRKCA 11/4885PRKCB 6/4885PRKCE 16/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.