SCHEMBL29375545

SCHEMBL29375545

O=[N+]([O-])c1ccc2c(cnn2C2COC2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLS O94925 1/20 0.50
SLC6A2 P23975 1/20 0.40
MAPT P10636 5/20 0.38
POLB P06746 2/20 0.38
NOS1 P29475 2/20 0.38
MAOB P27338 1/20 0.38
ALDH1A1 P00352 4/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38
KDR P35968 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CYP3A4 P08684 2/20 0.37
HTR3E A5X5Y0 1/20 0.37
HTR3B O95264 1/20 0.37
SLC6A4 P31645 1/20 0.37
CYP2C19 P33261 1/20 0.37
THPO P40225 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27083893 1.00 GLS (0.50) GLSSLC6A2MAPTPOLBNOS1
SCHEMBL30448181 0.90 GLS (0.46) GLSSLC6A2MAPTPOLBNOS1
SCHEMBL31304459 0.87 GLS (0.53) GLSSLC6A2MAPTPOLBNOS1
SCHEMBL14910335 0.87 GLS (0.53) GLSSLC6A2MAPTPOLBNOS1
SCHEMBL15910780 0.85 GLS (0.51) GLSSLC6A2MAPTPOLBNOS1
SCHEMBL3354657 0.83 GLS (0.49) GLSSLC6A2MAPTPOLBNOS1
SCHEMBL3355202 0.81 GLS (0.50) GLSMAPTPOLBALDH1A1NPC1
SCHEMBL29377201 0.81 GLS (0.50) GLSMAPTPOLBALDH1A1NPC1
SCHEMBL3357246 0.79 MAPT (0.51) GLSMAPTPOLBALDH1A1CYP1A2
SCHEMBL3355498 0.78 GLS (0.47) GLSMAPTPOLBALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116322683-A Compounds as C5AR inhibitors 科越医药(苏州)有限公司 2023-06-23 CN disclosed
EP-4192816-A1 COMPOUNDS AS C5AR INHIBITORS Kira Pharmaceuticals (Suzhou) Ltd. (CN) 2023-06-14 EP disclosed
WO-2022028586-A1 COMPOUNDS AS C5AR INHIBITORS KIRA PHARMACEUTICALS (SUZHOU) LTD. (CN) 2022-02-10 WO disclosed