SCHEMBL29375615

SCHEMBL29375615

COc1ccc(COc2c(F)cc(C(=O)O)cc2C2SCCCS2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
NPC1 O15118 2/20 0.47
POLB P06746 1/20 0.47
PLA2G4B P0C869 1/20 0.43
TP53 P04637 1/20 0.41
PKM P14618 1/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
MRGPRX4 Q96LA9 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
PPARA Q07869 1/20 0.40
PTGER1 P34995 2/20 0.39
NR4A2 P43354 1/20 0.39
KDM5A P29375 1/20 0.39
KDM4C Q9H3R0 1/20 0.39
KDM5B Q9UGL1 1/20 0.39
FFAR1 O14842 4/20 0.38
HRH3 Q9Y5N1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22466074 1.00 RAB9A (0.47) RAB9ASMN1; SMN2NPC1POLBPLA2G4B
SCHEMBL30903838 0.96 RAB9A (0.49) RAB9ASMN1; SMN2NPC1POLBPLA2G4B
SCHEMBL22465913 0.88 MEN1 (0.45) MRGPRX4PTGER1NR4A2
SCHEMBL29375274 0.88 MEN1 (0.45) MRGPRX4PTGER1NR4A2
SCHEMBL30903834 0.84 MEN1 (0.47) RAB9ASMN1; SMN2NPC1MRGPRX4PTGER1
SCHEMBL22466085 0.83 SENP5 (0.46) RAB9ASMN1; SMN2NPC1TP53RXFP1
SCHEMBL29378052 0.83 SENP5 (0.46) RAB9ASMN1; SMN2NPC1TP53RXFP1
SCHEMBL22468980 0.83 RAB9A (0.45) RAB9ASMN1; SMN2NPC1POLBPLA2G4B
SCHEMBL22465887 0.83 MAOB (0.37) RAB9ANPC1
SCHEMBL22466141 0.83 MAOB (0.37) ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114025847-B Compounds and compositions as modulators of TLR signaling 神经孔疗法股份有限公司 2024-05-24 CN disclosed
EP-3946599-A1 COMPOUNDS AND COMPOSITIONS AS MODULATORS OF TLR SIGNALING Neuropore Therapies, Inc. (US) 2022-02-09 EP disclosed
CN-114025847-A Compounds and compositions as modulators of TLR signaling 神经孔疗法股份有限公司 2022-02-08 CN disclosed