SCHEMBL29375779

SCHEMBL29375779

CC(=O)Nc1ccc(N)c2c1CCCC2=O

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BAZ2B Q9UIF8 1/20 0.40
MAPT P10636 3/20 0.40
HDAC3 O15379 2/20 0.39
HDAC1 Q13547 2/20 0.39
HDAC2 Q92769 2/20 0.39
BRD4 O60885 3/20 0.37
NPC1 O15118 3/20 0.37
ALDH1A1 P00352 3/20 0.37
HPGD P15428 2/20 0.37
RXFP1 Q9HBX9 1/20 0.36
RAB9A P51151 2/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
POLB P06746 1/20 0.35
KDM4E B2RXH2 2/20 0.35
ADRA2A P08913 1/20 0.34
MAOA P21397 1/20 0.34
PARP14 Q460N5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22463098 1.00 BAZ2B (0.40) BAZ2BMAPTHDAC3HDAC1HDAC2
SCHEMBL7652191 0.88 BAZ2B (0.44) BAZ2BMAPTBRD4NPC1ALDH1A1
SCHEMBL22519655 0.81 BRD4 (0.40) MAPTBRD4ALDH1A1HPGDKDM4E
SCHEMBL25692600 0.81 AAK1 (0.39) MAPTBRD4ALDH1A1HPGDRAB9A
SCHEMBL7653960 0.79 BAZ2B (0.42) BAZ2BMAPTBRD4NPC1ALDH1A1
SCHEMBL22463090 0.78 L3MBTL1 (0.40) BAZ2BMAPTBRD4ALDH1A1HPGD
SCHEMBL22463095 0.78 MAPT (0.45) BAZ2BMAPTALDH1A1HPGDPOLB
SCHEMBL29375798 0.78 MAPT (0.45) BAZ2BMAPTALDH1A1HPGDPOLB
SCHEMBL29376104 0.78 L3MBTL1 (0.40) BAZ2BMAPTBRD4ALDH1A1HPGD
SCHEMBL25692601 0.77 BAZ2B (0.36) BAZ2BMAPTBRD4ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117263948-B Compounds and conjugates thereof 免疫医疗有限公司 2024-11-22 CN disclosed
CN-118240003-A Compounds and conjugates thereof 免疫医疗有限公司 2024-06-25 CN disclosed
CN-118221763-A Compounds and conjugates thereof 免疫医疗有限公司 2024-06-21 CN disclosed
CN-113631196-B Compounds and conjugates thereof 免疫医疗有限公司 2024-03-15 CN disclosed
CN-117263948-A Compounds and conjugates thereof 免疫医疗有限公司 2023-12-22 CN disclosed
CN-116829592-A Therapeutic B7-H4 binding molecules 免疫医疗有限公司 2023-09-29 CN disclosed
EP-4211166-A1 THERAPEUTIC B7-H4 BINDING MOLECULES MedImmune Limited (GB) 2023-07-19 EP disclosed
EP-4093439-A1 COMPOUNDS AND CONJUGATES THEREOF MedImmune Limited (GB) 2022-11-30 EP disclosed
CN-114980934-A Compounds and conjugates thereof 免疫医疗有限公司 2022-08-30 CN disclosed
WO-2022053650-A1 THERAPEUTIC B7-H4 BINDING MOLECULES MEDIMMUNE LIMITED (GB) 2022-03-17 WO disclosed
EP-3946464-A1 COMPOUNDS AND CONJUGATES THEREOF MedImmune Limited (GB) 2022-02-09 EP disclosed