N,N-Hexamethyleneamiloride

N,N-Hexamethyleneamiloride

SCHEMBL29384339

N=C(N)NC(=O)c1nc(Cl)c(N2CCCCCC2)nc1N

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 15/20 0.62
SLC9A5 Q14940 2/20 0.62
LMNA P02545 2/20 0.62
NPC1 O15118 2/20 0.62
ALDH1A1 P00352 2/20 0.62
RAB9A P51151 2/20 0.62
MEN1 O00255 1/20 0.62
TP53 P04637 1/20 0.62
CYP1A2 P05177 1/20 0.62
CYP2D6 P10635 1/20 0.62
TSHR P16473 1/20 0.62
SLC9A1 P19634 1/20 0.62
ADORA2A P29274 1/20 0.62
ADORA2B P29275 1/20 0.62
CYP2C19 P33261 1/20 0.62
THPO P40225 1/20 0.62
PMP22 Q01453 1/20 0.62
KMT2A Q03164 1/20 0.62
KCNH2 Q12809 1/20 0.62
SCN5A Q14524 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11460538 1.00 PLAU (0.62) PLAUSLC9A5LMNANPC1ALDH1A1
N,N-Hexamethyleneamiloride SCHEMBL7862943 1.00 PLAU (0.62) PLAUSLC9A5LMNANPC1ALDH1A1
SCHEMBL11469206 0.99 PLAU (0.60) PLAUSLC9A5LMNANPC1ALDH1A1
SCHEMBL26104614 0.88 ALDH1A1 (0.47) PLAUSLC9A5LMNANPC1ALDH1A1
SCHEMBL11615921 0.85 PLAU (0.53) PLAUSLC9A5LMNANPC1ALDH1A1
SCHEMBL15082596 0.84 PLAU (0.57) PLAUSLC9A5LMNANPC1ALDH1A1
Amiloride SCHEMBL365969 0.82 SCNN1A (0.55) PLAUSLC9A5LMNANPC1ALDH1A1
SCHEMBL17704667 0.82 PLAU (0.62) PLAUSLC9A5LMNANPC1ALDH1A1
SCHEMBL11467427 0.80 GRM5 (0.48) PLAUSLC9A5LMNANPC1ALDH1A1
SCHEMBL26106945 0.80 GRM5 (0.58) PLAUSLC9A5LMNANPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4577202-A1 USE OF A THERAPEUTIC AGENT WITH SODIUM-HYDROGEN ANTIPORTER 1 INHIBITORY ACTIVITY FOR THE TREATMENT AND PREVENTION OF DISEASES ASSOCIATED WITH CHRONIC FATIGUE, EXHAUSTION AND/OR EXERTIONAL INTOLERANCE Mitodicure GmbH (DE) 2025-07-02 EP claimed
CN-119923254-A Use of therapeutic agents having sodium hydrogen antiport 1 inhibitory activity for the treatment and prevention of diseases associated with chronic fatigue, exhaustion and/or fatigue intolerance 米托迪治愈有限责任公司 2025-05-02 CN claimed
WO-2024042160-A1 USE OF A THERAPEUTIC AGENT WITH SODIUM-HYDROGEN ANTIPORTER 1 INHIBITORY ACTIVITY FOR THE TREATMENT AND PREVENTION OF DISEASES ASSOCIATED WITH CHRONIC FATIGUE, EXHAUSTION AND/OR EXERTIONAL INTOLERANCE MITODICURE GMBH (DE) 2024-02-29 WO claimed
CN-117323334-A Application of NHE1 inhibitor in preparation of medicine for preventing and treating multiple myeloma 暨南大学 2024-01-02 CN claimed
CN-114712361-A Compositions and methods for preventing or reducing the incidence of transient ischemic attacks 莫尔豪斯医学院 2022-07-08 CN claimed
CN-109475552-B Methods and compositions for appetite control and weight management 上海药苑生物科技有限公司 2022-04-05 CN claimed
EP-4577202-A1 USE OF A THERAPEUTIC AGENT WITH SODIUM-HYDROGEN ANTIPORTER 1 INHIBITORY ACTIVITY FOR THE TREATMENT AND PREVENTION OF DISEASES ASSOCIATED WITH CHRONIC FATIGUE, EXHAUSTION AND/OR EXERTIONAL INTOLERANCE Mitodicure GmbH (DE) 2025-07-02 EP disclosed
CN-119923254-A Use of therapeutic agents having sodium hydrogen antiport 1 inhibitory activity for the treatment and prevention of diseases associated with chronic fatigue, exhaustion and/or fatigue intolerance 米托迪治愈有限责任公司 2025-05-02 CN disclosed
EP-4536354-A1 MINOXIDIL ADJUVANT THERAPIES Jupiter Wellness, Inc. (US) 2025-04-16 EP disclosed
CN-110742891-B Composition for reducing damage to nervous system, method for producing the same, and use of the same 莫尔豪斯医学院 2024-04-05 CN disclosed
WO-2024042160-A1 USE OF A THERAPEUTIC AGENT WITH SODIUM-HYDROGEN ANTIPORTER 1 INHIBITORY ACTIVITY FOR THE TREATMENT AND PREVENTION OF DISEASES ASSOCIATED WITH CHRONIC FATIGUE, EXHAUSTION AND/OR EXERTIONAL INTOLERANCE MITODICURE GMBH (DE) 2024-02-29 WO disclosed
CN-117323334-A Application of NHE1 inhibitor in preparation of medicine for preventing and treating multiple myeloma 暨南大学 2024-01-02 CN disclosed
CN-117243839-A Minoxidil adjuvant therapy 应用生物学股份有限公司 2023-12-19 CN disclosed
CN-114712361-A Compositions and methods for preventing or reducing the incidence of transient ischemic attacks 莫尔豪斯医学院 2022-07-08 CN disclosed
CN-109475552-B Methods and compositions for appetite control and weight management 上海药苑生物科技有限公司 2022-04-05 CN disclosed
US-20220040225-A1 METHOD OF ADMINISTRATION AND TREATMENT DYVE BIOSCIENCES, INC. 2022-02-10 US disclosed