SCHEMBL29389889

SCHEMBL29389889

NC(=O)c1c(F)cccc1Nc1nc(Cl)ncc1Br

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.47
BCR P11274 1/20 0.47
IGF1R P08069 3/20 0.42
MAPK8 P45983 4/20 0.42
MAPK9 P45984 2/20 0.42
MAPK10 P53779 2/20 0.42
MAPT P10636 2/20 0.41
HTT P42858 1/20 0.41
JAK2 O60674 2/20 0.40
AURKA O14965 1/20 0.40
AURKB Q96GD4 1/20 0.40
PIM1 P11309 2/20 0.40
JAK3 P52333 2/20 0.40
CDC7 O00311 1/20 0.40
DAPK3 O43293 1/20 0.40
ROCK2 O75116 1/20 0.40
PRKD3 O94806 1/20 0.40
MAP4K4 O95819 1/20 0.40
PAK4 O96013 1/20 0.40
PRKACA P17612 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22500906 1.00 ABL1 (0.47) ABL1BCRIGF1RMAPK8MAPK9
SCHEMBL1204114 0.88 MAPK10 (0.49) ABL1BCRIGF1RMAPK8MAPK9
SCHEMBL22521033 0.87 MAPK8 (0.43) ABL1BCRIGF1RMAPK8MAPK9
SCHEMBL30833652 0.78 IGF1R (0.40) ABL1BCRIGF1RMAPK8MAPK9
SCHEMBL22520850 0.78 AURKA (0.57) ABL1IGF1RMAPK8MAPK9MAPK10
SCHEMBL22520990 0.77 CDK5 (0.47) IGF1RMAPK8MAPK9MAPK10JAK2
SCHEMBL29172717 0.77 ZAP70 (0.49) IGF1RMAPK8MAPK9MAPK10JAK2
SCHEMBL22520852 0.76 MAPK8 (0.48) IGF1RMAPK8MAPK9MAPK10JAK2
SCHEMBL29526063 0.75 MAPK10 (0.47) IGF1RMAPK8MAPK9MAPK10JAK2
SCHEMBL27166361 0.75 CDK5 (0.52) IGF1RMAPK8MAPK9MAPK10JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250136619-A1 HETEROBIFUNCTIONAL COMPOUNDS AND THEIR USE IN TREATING DISEASE HALDA THERAPEUTICS OPCO, INC. 2025-05-01 US disclosed
CN-117715904-A CDK2 degrading agents and uses thereof 凯麦拉医疗公司 2024-03-15 CN disclosed
WO-2024054602-A1 HETEROBIFUNCTIONAL COMPOUNDS AND METHODS OF TREATING DISEASE HALDA THERAPEUTICS OPCO, INC. (US) 2024-03-14 WO disclosed
EP-4334307-A1 CDK2 DEGRADERS AND USES THEREOF Kymera Therapeutics, Inc. (US) 2024-03-13 EP disclosed
WO-2023059583-A1 HETEROBIFUNCTIONAL COMPOUNDS AND THEIR USE IN TREATING DISEASE HALDA THERAPEUTICS OPCO, INC. (US) 2023-04-13 WO disclosed
WO-2023059581-A1 HETEROBIFUNCTIONAL COMPOUNDS AND THEIR USE IN TREATING DISEASE HALDA THERAPEUTICS OPCO, INC. (US) 2023-04-13 WO disclosed
WO-2022236058-A1 CDK2 DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS, INC. (US) 2022-11-10 WO disclosed
EP-3947368-A1 CDK2/5 DEGRADERS AND USES THEREOF Dana-Farber Cancer Institute, Inc. (US) 2022-02-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250136619-A1 HETEROBIFUNCTIONAL COMPOUNDS AND THEIR USE IN TREATING DISEASE CDK9, AURKB, AURKC ABL1 121/4885BCR 1074/4885IGF1R 1539/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.