SCHEMBL29392011

SCHEMBL29392011

COc1cc(OCCCN2CCN(C)CC2)cc2nc(Cl)c(C#N)c(Cl)c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIOK3 O14730 2/20 0.47
SRC P12931 12/20 0.44
KDR P35968 4/20 0.44
WEE2 P0C1S8 2/20 0.43
WEE1 P30291 2/20 0.43
PKMYT1 Q99640 2/20 0.43
FYN P06241 2/20 0.42
DRD3 P35462 2/20 0.42
HRH3 Q9Y5N1 2/20 0.42
STK25 O00506 1/20 0.42
CIT O14578 1/20 0.42
MAP2K7 O14733 1/20 0.42
CHEK1 O14757 1/20 0.42
CASK O14936 1/20 0.42
GAK O14976 1/20 0.42
EPHB6 O15197 1/20 0.42
MAP3K13 O43283 1/20 0.42
MAP3K7 O43318 1/20 0.42
RIPK2 O43353 1/20 0.42
NUAK1 O60285 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3194260 0.72 SRC (0.73) RIOK3SRCWEE2WEE1PKMYT1
SCHEMBL4489514 0.68 WEE2 (0.71) RIOK3SRCKDRWEE2WEE1
SCHEMBL4764821 0.68 SRC (0.51) RIOK3SRCKDRWEE2WEE1
SCHEMBL16827594 0.67 HRH3 (0.54) SRCFYNDRD3HRH3CHEK1
SCHEMBL16618011 0.66 LMNA (0.45) RIOK3SRCKDRWEE2WEE1
SCHEMBL30544811 0.66 SRC (0.57) RIOK3SRCKDRWEE2WEE1
SCHEMBL30326588 0.65 HRH3 (0.57) DRD3HRH3CHEK1HRH2SLC6A4
SCHEMBL12311793 0.65 HRH3 (0.60) DRD3HRH3DRD2SLC6A2HTR2A
SCHEMBL16747775 0.65 BRD4 (0.48) SRCKDRDRD3DRD2TERT
SCHEMBL2206979 0.65 HRH3 (0.59) DRD3HRH3DRD2SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902029-B2 CRYSTALLINE FORMS OF 4-[(2,4-DICHLORO-5-METHOXYPHENYL)AMINO]-6-METHOXY-7-[3-(4-METHYL-1-PIPERAZINYL)PROPOXY]-3-QUINOLINECARB-ONITRILE AND METHODS OF PREPARING THE SAME WYETH LLC (US) 2022-02-16 EP disclosed