SCHEMBL2939477

SCHEMBL2939477

CCCNC(=O)c1ccccc1Nc1nc(Cl)ncc1Cl.CCCNC(=O)c1ccccc1Nc1nc(Nc2ccc3c(c2)C(C)(C)CCC(=O)N3)ncc1Cl

nearest known ligand 0.77

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MET P08581 19/20 0.77
INSR P06213 11/20 0.77
ALK Q9UM73 7/20 0.47
ULK1 O75385 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL886640 0.97 MET (0.82) METINSRALKULK1
SCHEMBL886145 0.93 MET (0.80) METINSRALKULK1
SCHEMBL886710 0.87 MET (1.00) METINSRALKULK1
SCHEMBL886159 0.84 MET (0.74) METINSRALKULK1
SCHEMBL3009983 0.84 MET (0.61) METINSRALKULK1
SCHEMBL2942745 0.82 MET (0.77) METINSRALKULK1
SCHEMBL2062335 0.82 MET (0.78) METINSR
SCHEMBL2061757 0.81 MET (0.85) METINSR
SCHEMBL886731 0.80 MET (0.74) METINSRALKULK1
SCHEMBL885994 0.79 MET (0.73) METINSRALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222647-A1 FUSED BICYCLIC DERIVATIVES OF 2,4-DIAMINOPYRIMIDINE AS ALK AND C-MET INHIBITORS Cephalon, Inc. (US) 2010-09-01 EP disclosed
WO-2008051547-A1 FUSED BICYCLIC DERIVATIVES OF 2,4-DIAMINOPYRIMIDINE AS ALK AND C-MET INHIBITORS CEPHALON, INC. (US) 2008-05-02 WO disclosed