SCHEMBL29404355

SCHEMBL29404355

CCc1cc(Cl)nnc1Cl

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.44
CTRC Q99895 1/20 0.34
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
GRIN2B Q13224 1/20 0.32
GRIN2C Q14957 1/20 0.32
GRIN3A Q8TCU5 1/20 0.32
ALDH1A1 P00352 4/20 0.32
CASP1 P29466 1/20 0.32
LMNA P02545 1/20 0.32
PKM P14618 1/20 0.32
RAB9A P51151 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1188816 1.00 TDP1 (0.44) TDP1CTRCGRIN2DGRIN3BGRIN1
SCHEMBL30500471 0.82 TDP1 (0.41) TDP1ALDH1A1PKM
SCHEMBL7832945 0.82 TDP1 (0.41) TDP1ALDH1A1PKM
SCHEMBL16454767 0.79 GRIN2D (0.35) CTRCGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL2259889 0.79 TDP1 (0.33) TDP1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL1268563 0.79 TDP1 (0.39) TDP1CTRCRAB9A
SCHEMBL29993398 0.77 TDP1 (0.41) TDP1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL3024535 0.77 TDP1 (0.41) TDP1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL3012650 0.77 NOS3 (0.39) TDP1CTRCGRIN2DGRIN3BGRIN1
SCHEMBL5567705 0.77 TDP1 (0.38) TDP1CTRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119300833-A Novel compounds 豪夫迈·罗氏有限公司 2025-01-10 CN disclosed
CN-118265701-A Pyridazine derivatives as inhibitors of NLRP3 豪夫迈·罗氏有限公司 2024-06-28 CN disclosed
CN-114072390-B RAD51 inhibitors 赛泰尔治疗公司 2024-06-11 CN disclosed
CN-111566089-B IRE1 small molecule inhibitors 康奈尔大学 2023-11-17 CN disclosed
CN-114072390-A RAD51 inhibitors 赛泰尔治疗公司 2022-02-18 CN disclosed