SCHEMBL29410004

SCHEMBL29410004

COC(=O)c1ncc(Cl)nc1N

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.45
KDM4E B2RXH2 6/20 0.42
PKM P14618 3/20 0.42
ALDH1A1 P00352 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
GRM5 P41594 2/20 0.42
MAPKAPK2 P49137 7/20 0.40
PIK3CD O00329 1/20 0.40
RCE1 Q9Y256 1/20 0.40
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TSHR P16473 1/20 0.38
ABL1 P00519 1/20 0.37
MAPK1 P28482 1/20 0.37
GLA P06280 1/20 0.37
GAA P10253 1/20 0.37
PLAU P00749 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL260853 1.00 NPSR1 (0.45) NPSR1KDM4EPKMALDH1A1SMN1; SMN2
SCHEMBL29844710 0.88 GRM5 (0.52) NPSR1KDM4EPKMALDH1A1SMN1; SMN2
SCHEMBL261816 0.88 GRM5 (0.52) NPSR1KDM4EPKMALDH1A1SMN1; SMN2
SCHEMBL20046668 0.84 NPSR1 (0.56) NPSR1KDM4EPKMALDH1A1SMN1; SMN2
SCHEMBL1680511 0.82 PLAU (0.53) NPSR1KDM4EPKMALDH1A1SMN1; SMN2
SCHEMBL4014560 0.82 NPSR1 (0.48) NPSR1KDM4EPKMALDH1A1SMN1; SMN2
SCHEMBL29585697 0.82 NPSR1 (0.48) NPSR1KDM4EPKMALDH1A1SMN1; SMN2
SCHEMBL25399004 0.81 NPSR1 (0.47) NPSR1KDM4EPKMALDH1A1SMN1; SMN2
SCHEMBL361753 0.81 NPSR1 (0.47) NPSR1KDM4EPKMALDH1A1SMN1; SMN2
SCHEMBL12248189 0.81 NPSR1 (0.47) NPSR1KDM4EPKMALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3968983-A1 MACROCYCLIC BROAD SPECTRUM ANTIBIOTICS F. Hoffmann-La Roche AG (CH) 2022-03-23 EP disclosed