SCHEMBL29411908

SCHEMBL29411908

COCCOc1ccc(Nc2ncc(F)c(Nc3ccc(C(=O)NN)cc3)n2)cc1

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EGFR P00533 8/20 0.65
BTK Q06187 3/20 0.65
ITK Q08881 3/20 0.65
JAK2 O60674 1/20 0.65
LYN P07948 1/20 0.65
TEC P42680 1/20 0.65
TXK P42681 1/20 0.65
BMX P51813 1/20 0.65
JAK3 P52333 1/20 0.65
CD69 Q07108 1/20 0.65
SYK P43405 6/20 0.65
AURKA O14965 6/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28704339 1.00 EGFR (0.65) EGFRBTKITKJAK2LYN
SCHEMBL28720308 0.92 EGFR (0.65) EGFRBTKITKJAK2LYN
SCHEMBL29411905 0.91 EGFR (0.66) EGFRBTKITKJAK2LYN
SCHEMBL28704792 0.91 EGFR (0.66) EGFRBTKITKJAK2LYN
SCHEMBL28718244 0.90 EGFR (0.72) EGFRBTKITKJAK2LYN
SCHEMBL29411924 0.90 EGFR (0.72) EGFRBTKITKJAK2LYN
SCHEMBL22909543 0.87 SYK (0.69) EGFRBTKITKJAK2LYN
SCHEMBL29412027 0.85 BTK (0.65) EGFRBTKITKJAK2LYN
SCHEMBL28715173 0.85 BTK (0.65) EGFRBTKITKJAK2LYN
SCHEMBL23409017 0.85 SYK (0.68) EGFRBTKITKJAK2LYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114181159-A Hydrazide derivative containing 2,4, 5-trisubstituted pyrimidine, preparation method and application thereof 南通大学 2022-03-15 CN claimed
CN-114181159-B 2,4, 5-trisubstituted pyrimidine hydrazide derivative and preparation method and application thereof 南通大学 2024-02-20 CN disclosed
CN-114181159-A Hydrazide derivative containing 2,4, 5-trisubstituted pyrimidine, preparation method and application thereof 南通大学 2022-03-15 CN disclosed