SCHEMBL29417293

SCHEMBL29417293

CC(C)(C)C(=O)NCc1ccc(F)c(C#N)c1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGES O14684 5/20 0.50
HDAC6 Q9UBN7 1/20 0.47
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA7 P43166 1/20 0.46
CA14 Q9ULX7 1/20 0.46
CNR2 P34972 1/20 0.45
SMO Q99835 1/20 0.45
CHRNA7 P36544 1/20 0.43
CACNA1H O95180 1/20 0.43
AR P10275 1/20 0.41
IMPDH2 P12268 1/20 0.40
VNN1 O95497 1/20 0.40
EPHX2 P34913 1/20 0.40
NR1H4 Q96RI1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18810055 1.00 PTGES (0.50) PTGESHDAC6CA1CA2CA7
SCHEMBL18809962 0.83 PTGES (0.48) PTGESHDAC6CA1CA2CA7
SCHEMBL3359490 0.81 CYP2C9 (0.50) CHRNA7CACNA1HVNN1
SCHEMBL18809969 0.81 ERCC1 (0.55) PTGESSMOCHRNA7CACNA1HAR
SCHEMBL29417087 0.81 ERCC1 (0.55) PTGESSMOCHRNA7CACNA1HAR
SCHEMBL25590873 0.78 HDAC6 (0.50) PTGESHDAC6CA1CA2CA7
SCHEMBL25489342 0.78 CACNA1H (0.39) CHRNA7CACNA1HARVNN1
SCHEMBL25488907 0.77 LOXL2 (0.50) CHRNA7CACNA1HARVNN1
SCHEMBL29417203 0.76 PTGES (0.46) PTGESCHRNA7CACNA1HVNN1
SCHEMBL18809824 0.76 PTGES (0.46) PTGESCHRNA7CACNA1HVNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137513-B Pyrimidine derivatives ASKA 制药株式会社 2022-03-01 CN disclosed