SCHEMBL29424797

SCHEMBL29424797

COc1ccnc2[nH]ccc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.60
PRKCI P41743 3/20 0.53
AXL P30530 1/20 0.53
AURKB Q96GD4 3/20 0.47
IKBKB O14920 1/20 0.47
CHUK O15111 1/20 0.47
DAPK3 O43293 1/20 0.47
JAK2 O60674 1/20 0.47
PRKD3 O94806 1/20 0.47
MAP4K4 O95819 1/20 0.47
PAK4 O96013 1/20 0.47
CSF1R P07333 1/20 0.47
RET P07949 1/20 0.47
IGF1R P08069 1/20 0.47
FGFR1 P11362 1/20 0.47
PRKACA P17612 1/20 0.47
FLT1 P17948 1/20 0.47
LTK P29376 1/20 0.47
GRK5 P34947 1/20 0.47
KDR P35968 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL298491 1.00 BRD4 (0.60) BRD4PRKCIAXLAURKBIKBKB
SCHEMBL30669883 0.84 BRD4 (0.52) BRD4PRKCIAXLAURKBIKBKB
SCHEMBL2992617 0.81 NUDT1 (0.55) BRD4PRKCIAXLAURKBIKBKB
SCHEMBL12605521 0.81 CCNK (0.51) BRD4PRKCIAXLAURKBIKBKB
SCHEMBL2986157 0.80 CIT (0.50) BRD4PRKCIAXLAURKBIKBKB
SCHEMBL30461709 0.79 NUDT1 (0.52) BRD4PRKCIAXLAURKBIKBKB
SCHEMBL2988049 0.79 NUDT1 (0.52) BRD4PRKCIAXLAURKBIKBKB
SCHEMBL10125070 0.79 BRD4 (0.66) BRD4PRKCIAURKBIKBKBCHUK
SCHEMBL858602 0.79 BRD4 (0.62) BRD4PRKCIAURKBIKBKBCHUK
SCHEMBL29120136 0.78 PRKCI (0.50) BRD4PRKCIAXLAURKBIKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118974044-A Compounds of formula (I) 赛洛私人有限公司 2024-11-15 CN disclosed
US-20240034799-A1 METHODS AND SYSTEMS OF STRATIFYING INFLAMMATORY DISEASE PATIENTS CEDARS SINAI MEDICAL CENTER (US) 2024-02-01 US disclosed
US-20230279491-A1 TREATMENTS FOR A SUB-POPULATION OF INFLAMMATORY BOWEL DISEASE PATIENTS CEDARS-SINAI MEDICAL CENTER 2023-09-07 US disclosed
CN-114746090-A Azaindole carboxamide compounds for the treatment of mycobacterial infections 结核病药物开发全球联盟公司 2022-07-12 CN disclosed
CN-114040915-A Bicyclic heteroaryl derivatives as ectonucleotide pyrophosphatase phosphodiesterase 1 inhibitors 里伯赛恩斯有限责任公司 2022-02-11 CN disclosed