SCHEMBL2943049

SCHEMBL2943049

COc1ccc(Sc2nc(N)nc3c2ncn3CC2(O[C](COC(=O)OC(C)(C)C)COC(=O)OC(C)(C)C)CC2)cc1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.34
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
ADORA2A P29274 1/20 0.33
HK1 P19367 1/20 0.32
HKDC1 Q2TB90 1/20 0.32
DHFR P00374 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
CYP1A2 P05177 2/20 0.31
SLC29A1 Q99808 1/20 0.31
CNR2 P34972 1/20 0.30
ALDH1A1 P00352 1/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2941709 0.89 HK1 (0.35) CYP2C19HSP90AA1HSP90AB1ADORA2AHK1
SCHEMBL2937081 0.89 HSP90AA1 (0.33) CYP2C19HSP90AA1HSP90AB1ADORA2AHK1
SCHEMBL2913792 0.85 HSP90AA1 (0.32) CYP2C19HSP90AA1HSP90AB1ADORA2AHK1
SCHEMBL4275862 0.85 HK1 (0.33) CYP2C19HSP90AA1HSP90AB1ADORA2AHK1
SCHEMBL2995160 0.83 ADORA2A (0.35) CYP2C19HSP90AA1HSP90AB1ADORA2AHK1
SCHEMBL2939394 0.82 CDK1 (0.32) CYP2C19
SCHEMBL2936424 0.79 HK1 (0.34) CYP2C19HSP90AA1HSP90AB1ADORA2AHK1
SCHEMBL2937343 0.78 CYP1A2 (0.36) CYP2C19ADORA2ACYP1A2SLC29A1
SCHEMBL4268504 0.78 HK1 (0.32) CYP2C19HSP90AA1HSP90AB1ADORA2AHK1
SCHEMBL2914520 0.78 HSP90AA1 (0.31) CYP2C19HSP90AA1HSP90AB1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1358198-B1 NOVEL ACYCLIC NUCLEOSIDE PHOSPHONATE DERIVATIVES, SALTS THEREOF AND PROCESS FOR THE PREPARATION OF THE SAME LG LIFE SCIENCES LTD (KR) 2010-08-25 EP claimed