SCHEMBL29437964

SCHEMBL29437964

CCC1(CC)OCc2cccc(Oc3ccc(N4C(=O)N[C@](C)(CC)C4=O)cn3)c21

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.35
MCOLN3 Q8TDD5 1/20 0.35
MMP13 P45452 2/20 0.33
ELANE P08246 1/20 0.31
AR P10275 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15303437 1.00 KDM4E (0.35) KDM4EMCOLN3MMP13ELANEAR
SCHEMBL30939625 0.93 KDM4E (0.35) KDM4EMCOLN3MMP13ELANEAR
SCHEMBL9904969 0.93 KDM4E (0.35) KDM4EMCOLN3MMP13ELANEAR
SCHEMBL15303543 0.86 KDM4E (0.38) KDM4EMCOLN3MMP13
SCHEMBL9924311 0.86 KDM4E (0.34) KDM4EMCOLN3MMP13
SCHEMBL30939527 0.86 KDM4E (0.34) KDM4EMCOLN3MMP13
SCHEMBL21116329 0.83 AR (0.39) KDM4EMCOLN3MMP13ELANEAR
SCHEMBL17180633 0.82 KDM4E (0.35) KDM4EMCOLN3
SCHEMBL30939589 0.81 MMP13 (0.36) MMP13ELANEAR
SCHEMBL14158671 0.81 MMP13 (0.36) MMP13ELANEAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118267386-A Modulators of KV3 channels for the treatment of pain 奥提芙尼治疗学有限公司 2024-07-02 CN disclosed
CN-108472288-B Modulators of KV3 channels for the treatment of pain 奥提芙尼治疗学有限公司 2024-05-28 CN disclosed
US-11583527-B2 Hydantoin derivatives useful as Kv3 inhibitors AUTIFONY THERAPEUTICS LIMITED (GB) 2023-02-21 US disclosed
US-20220054490-A1 HYDANTOIN DERIVATIVES USEFUL AS KV3 INHIBITORS AUTIFONY THERAPEUTICS LIMITED (GB) 2022-02-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11583527-B2 Hydantoin derivatives useful as Kv3 inhibitors KCNN3, KCND3, KCNA3 KDM4E 1460/4885MCOLN3 288/4885MMP13 3782/4885
US-20220054490-A1 HYDANTOIN DERIVATIVES USEFUL AS KV3 INHIBITORS KCNN3, KCND3, KCNA3 KDM4E 1460/4885MCOLN3 288/4885MMP13 3782/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.