SCHEMBL29439677

SCHEMBL29439677

Sc1ncnc2nc(-c3cccc(I)c3)sc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.33
METAP2 P50579 1/20 0.32
EGFR P00533 1/20 0.32
IGF1R P08069 1/20 0.32
SRC P12931 1/20 0.32
KDR P35968 1/20 0.32
EPHB4 P54760 1/20 0.32
TYK2 P29597 1/20 0.32
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
PTPRF P10586 1/20 0.30
PTPN2 P17706 1/20 0.30
PTPN1 P18031 1/20 0.30
PIK3CG P48736 1/20 0.30
RAB9A P51151 3/20 0.30
KDM4E B2RXH2 2/20 0.30
NPC1 O15118 2/20 0.30
ALDH1A1 P00352 2/20 0.30
MAPT P10636 2/20 0.30
NFKB1 P19838 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22715176 1.00 IKBKB (0.33) IKBKBMETAP2EGFRIGF1RSRC
SCHEMBL29439756 0.86 IKBKB (0.44) IKBKBPIK3CGRAB9AKDM4ENPC1
SCHEMBL22715917 0.86 IKBKB (0.44) IKBKBPIK3CGRAB9AKDM4ENPC1
SCHEMBL22715327 0.82 CDC7 (0.35) IKBKBMETAP2EGFRIGF1RSRC
SCHEMBL29439823 0.82 CDC7 (0.35) IKBKBMETAP2EGFRIGF1RSRC
SCHEMBL22715521 0.79 LIMK1 (0.35) EGFRTYK2RAB9ANPC1
SCHEMBL29439774 0.79 LIMK1 (0.35) EGFRTYK2RAB9ANPC1
SCHEMBL793594 0.74 TYK2 (0.54) EGFRSRCTYK2
SCHEMBL23172713 0.71 RAB9A (0.40) RAB9AKDM4ENPC1ALDH1A1MAPT
SCHEMBL22715976 0.70 PIK3CG (0.59) IKBKBKDRPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118908957-A Small molecule inhibitors of NF- κB induced kinase 詹森药业有限公司 2024-11-08 CN disclosed
CN-114222737-B Small molecule inhibitors of NF- κB induced kinase 詹森药业有限公司 2024-07-26 CN disclosed
EP-3976597-A1 SMALL MOLECULE INHIBITORS OF NF-KB INDUCING KINASE Janssen Pharmaceutica NV (BE) 2022-04-06 EP disclosed
CN-114222737-A Small molecule inhibitor of NF-kB induced kinase 詹森药业有限公司 2022-03-22 CN disclosed