SCHEMBL29439730

SCHEMBL29439730

Nc1nc(C2CC2)nc2ccc(Cl)nc12

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 2/20 0.45
PDE8B O95263 12/20 0.43
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
HSD17B10 Q99714 1/20 0.41
NCOA3 Q9Y6Q9 1/20 0.41
DHFR P00374 2/20 0.33
MAP4K4 O95819 1/20 0.33
ACHE P22303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22715592 1.00 PDE10A (0.45) PDE10APDE8BKDM4ELMNAMAPT
SCHEMBL29439675 0.74 DHFR (0.53) DHFRMAP4K4
SCHEMBL3922711 0.74 DHFR (0.53) DHFRMAP4K4
SCHEMBL4095470 0.73 ACHE (0.35) HSD17B10DHFRMAP4K4ACHE
SCHEMBL15265691 0.73 PRMT5 (0.42) PDE10APDE8BKDM4ELMNAMAPT
SCHEMBL22715815 0.72 DHFR (0.36) HTTDHFRMAP4K4
SCHEMBL22715191 0.72 ADORA1 (0.41) KDM4EMAPTHTTDHFRMAP4K4
SCHEMBL22744486 0.72 DHFR (0.36) DHFRMAP4K4
SCHEMBL29439784 0.72 ADORA1 (0.41) KDM4EMAPTHTTDHFRMAP4K4
SCHEMBL22715906 0.72 DHFR (0.37) DHFRMAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118908957-A Small molecule inhibitors of NF- κB induced kinase 詹森药业有限公司 2024-11-08 CN disclosed
CN-114222737-B Small molecule inhibitors of NF- κB induced kinase 詹森药业有限公司 2024-07-26 CN disclosed
EP-3976597-A1 SMALL MOLECULE INHIBITORS OF NF-KB INDUCING KINASE Janssen Pharmaceutica NV (BE) 2022-04-06 EP disclosed
CN-114222737-A Small molecule inhibitor of NF-kB induced kinase 詹森药业有限公司 2022-03-22 CN disclosed