SCHEMBL29447286

SCHEMBL29447286

CC(C)(C)OC(=O)n1nc(I)c2cc(C=O)ccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K4 P45985 1/20 0.40
GABRG2 P18507 3/20 0.38
GABRB3 P28472 3/20 0.38
GABRA5 P31644 3/20 0.38
PTGER4 P35408 4/20 0.34
GABRA1 P14867 2/20 0.32
NR1H2 P55055 1/20 0.32
GABRA2 P47869 1/20 0.32
GABRA6 Q16445 1/20 0.32
HDAC1 Q13547 1/20 0.32
CYP2A6 P11509 1/20 0.32
HTR6 P50406 1/20 0.32
FAAH O00519 1/20 0.32
ELANE P08246 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
ROCK2 O75116 1/20 0.30
CHEK2 O96017 1/20 0.30
PRKACA P17612 1/20 0.30
RPS6KA3 P51812 1/20 0.30
PAK1 Q13153 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29951391 0.90 GABRG2 (0.36) MAP2K4GABRG2GABRB3GABRA5GABRA1
SCHEMBL9951845 0.85 MAP2K4 (0.40) MAP2K4GABRG2GABRB3GABRA5PTGER4
SCHEMBL14739081 0.83 HTR6 (0.46) MAP2K4GABRG2GABRB3GABRA5GABRA1
SCHEMBL9952523 0.83 MAP2K4 (0.42) MAP2K4GABRG2GABRB3GABRA5GABRA1
SCHEMBL24738080 0.82 GABRG2 (0.45) MAP2K4GABRG2GABRB3GABRA5GABRA1
SCHEMBL15169674 0.82 MAP2K4 (0.43) MAP2K4GABRG2GABRB3GABRA5GABRA1
SCHEMBL3514381 0.82 MAP2K4 (0.43) MAP2K4GABRG2GABRB3GABRA5GABRA1
SCHEMBL2732559 0.82 CDK1 (0.43) MAP2K4GABRG2GABRB3GABRA5ELANE
SCHEMBL5384350 0.81 MAP2K4 (0.38) MAP2K4GABRG2GABRB3GABRA5PTGER4
SCHEMBL5952597 0.81 ELANE (0.41) MAP2K4GABRG2GABRB3GABRA5ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112566905-B Substituted phenylpropenyl pyridine derivatives, preparation method and medical application thereof 上海海雁医药科技有限公司 2024-07-30 CN disclosed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
EP-3967687-A1 SUBSTITUTED PHENYLPROPENYLPYRIDINE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF Shanghai Haiyan Pharmaceutical Technology Co., Ltd (CN) 2022-03-16 EP disclosed