SCHEMBL29448796

SCHEMBL29448796

CC(C)(C)OC(=O)Nc1ccc(F)c(NC(=O)c2cccc(F)c2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.54
MEN1 O00255 5/20 0.54
MAPK14 Q16539 2/20 0.51
RAB9A P51151 7/20 0.49
NPC1 O15118 6/20 0.49
SMN1; SMN2 Q16637 4/20 0.49
KCNK3 O14649 2/20 0.49
KDM4E B2RXH2 1/20 0.49
CASP3 P42574 1/20 0.49
SENP7 Q9BQF6 1/20 0.49
SENP6 Q9GZR1 1/20 0.49
KCNK9 Q9NPC2 1/20 0.49
LMNA P02545 1/20 0.48
KCNQ3 O43525 1/20 0.46
KCNQ2 O43526 1/20 0.46
KCNE1 P15382 1/20 0.46
KCNQ1 P51787 1/20 0.46
NFKB1 P19838 1/20 0.46
HTT P42858 1/20 0.46
NFKB2 Q00653 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29286674 0.90 RAB9A (0.49) KMT2AMEN1MAPK14RAB9ANPC1
SCHEMBL29448759 0.90 RAB9A (0.49) KMT2AMEN1MAPK14RAB9ANPC1
SCHEMBL29448790 0.90 KCNK3 (0.51) KMT2AMEN1MAPK14RAB9ANPC1
SCHEMBL29448781 0.89 NPC1 (0.46) KMT2AMEN1MAPK14RAB9ANPC1
SCHEMBL7076019 0.88 NPC1 (0.60) KMT2AMEN1RAB9ANPC1SMN1; SMN2
SCHEMBL29448768 0.87 KCNQ3 (0.47) KMT2AMEN1MAPK14RAB9ANPC1
SCHEMBL20577799 0.87 RAB9A (0.47) KMT2AMEN1MAPK14RAB9ANPC1
SCHEMBL20578116 0.86 RAB9A (0.49) KMT2AMEN1MAPK14RAB9ANPC1
SCHEMBL20578151 0.86 SMN1; SMN2 (0.52) KMT2AMEN1MAPK14RAB9ANPC1
SCHEMBL29448809 0.85 BRAF (0.46) KMT2AMEN1MAPK14RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3412670-B1 PYRIDINE DERIVATIVES INHIBITING RAF KINASE AND VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR, PHARMACEUTICAL COMPOSITION CONTAINING THEM AND USE THEREOF SAMJIN PHARM CO LTD (KR) 2022-03-09 EP disclosed