SCHEMBL29450163

SCHEMBL29450163

CP(C)(=O)c1ccc(N)c(N)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.42
CYP3A4 P08684 3/20 0.42
ALOX15 P16050 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
TP53 P04637 1/20 0.42
THRB P10828 1/20 0.42
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
ALDH1A1 P00352 4/20 0.37
TSHR P16473 3/20 0.37
HPGD P15428 1/20 0.36
NR4A1 P22736 1/20 0.36
PKM P14618 2/20 0.33
MAPT P10636 2/20 0.33
KDM4E B2RXH2 1/20 0.33
GAA P10253 1/20 0.33
RAB9A P51151 1/20 0.33
HTR6 P50406 1/20 0.33
PTK2 Q05397 1/20 0.32
ESR1 P03372 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28724239 1.00 TDP1 (0.42) TDP1CYP3A4ALOX15SMN1; SMN2TP53
SCHEMBL1491739 0.82 CYP3A4 (0.48) TDP1CYP3A4ALOX15SMN1; SMN2TP53
SCHEMBL24073372 0.82 HPGD (0.33) TDP1CYP3A4ALOX15SMN1; SMN2TP53
SCHEMBL1491726 0.80 TSHR (0.46) TDP1CYP3A4ALOX15SMN1; SMN2TP53
SCHEMBL1491735 0.80 ALDH1A1 (0.46) ALDH1A1HPGD
SCHEMBL26602806 0.80 CA12 (0.44) TDP1CYP3A4ALDH1A1TSHRHPGD
SCHEMBL16995973 0.80 ALOX15 (0.46) TDP1CYP3A4ALOX15SMN1; SMN2THRB
SCHEMBL1491734 0.79 POLB (0.43) ALDH1A1HPGDMAPTGAAPOLB
SCHEMBL1491622 0.77 ALDH1A1 (0.52) TDP1CYP3A4SMN1; SMN2TP53THRB
SCHEMBL1491772 0.77 ALDH1A1 (0.53) TDP1CYP3A4THRBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116134025-B Amide phosphine oxide derivative and preparation method and application thereof 浙江海正药业股份有限公司 2025-04-04 CN disclosed
CN-114315899-B 3- (Aromatic ring imidazole) pyrazolopyrimidine derivative and application thereof 上海美迪西生物医药股份有限公司 2024-09-03 CN disclosed
CN-116134025-A Amide phosphine oxide derivative and preparation method and application thereof 浙江海正药业股份有限公司 2023-05-16 CN disclosed
CN-114315899-A 3- (aromatic benzimidazolyl) pyrazolopyrimidine derivative and application thereof 上海美迪西生物医药股份有限公司 2022-04-12 CN disclosed
WO-2022057858-A1 AMIDE PHOSPHINE OXIDE DERIVATIVE, PREPARATION METHOD THEREFOR, AND USE THEREOF 浙江海正药业股份有限公司 2022-03-24 WO disclosed