SCHEMBL29455649

SCHEMBL29455649

Cn1c(=O)oc2ccc(-c3ccc(CC(C#N)N=C(c4ccccc4)c4ccccc4)nn3)cc21

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 11/20 0.39
GPR55 Q9Y2T6 1/20 0.38
SCD5 Q86SK9 1/20 0.38
CTSC P53634 4/20 0.37
ALDH1A1 P00352 2/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25146985 1.00 KCNJ1 (0.39) KCNJ1GPR55SCD5CTSCALDH1A1
SCHEMBL24981827 0.87 KCNJ1 (0.43) KCNJ1GPR55SCD5CTSCALDH1A1
SCHEMBL24981577 0.85 KCNJ1 (0.51) KCNJ1GPR55SCD5CTSC
SCHEMBL24981584 0.82 KCNJ1 (0.45) KCNJ1GPR55SCD5CTSCALDH1A1
SCHEMBL24982008 0.81 KCNJ1 (0.43) KCNJ1GPR55SCD5CTSCALDH1A1
SCHEMBL31095717 0.81 CTSC (0.43) KCNJ1SCD5CTSCALDH1A1HPGD
SCHEMBL31095787 0.80 CTSC (0.39) GPR55SCD5CTSCALDH1A1HPGD
SCHEMBL31095604 0.80 CTSC (0.39) KCNJ1GPR55SCD5CTSCALDH1A1
SCHEMBL24982023 0.80 GPR55 (0.43) KCNJ1GPR55SCD5CTSC
SCHEMBL29455547 0.80 GPR55 (0.43) KCNJ1GPR55SCD5CTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022042591-A1 NITRILE DERIVATIVE THAT ACTS AS INHIBITOR OF DIPEPTIDYL PEPTIDASE 1 AND USE THEREOF 四川海思科制药有限公司 2022-03-03 WO disclosed