SCHEMBL29458221

SCHEMBL29458221

CN(C)CCOc1nc(N)ncc1C#N

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
CHEK1 O14757 1/20 0.36
CHEK2 O96017 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
TLR8 Q9NR97 1/20 0.35
CSNK1A1 P48729 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
CHRNB2 P17787 2/20 0.35
CHRNA4 P43681 2/20 0.35
NUDT1 P36639 1/20 0.35
HTR7 P34969 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25384842 1.00 ADORA2A (0.40) ADORA2AADORA1CHEK1CHEK2HRH3
SCHEMBL30509212 0.79 NOS1 (0.41) CHEK1CHEK2HTR7
SCHEMBL25382669 0.79 NOS1 (0.41) CHEK1CHEK2HTR7
SCHEMBL25383502 0.77 HTR7 (0.43) HRH3TLR8CHRNB2CHRNA4NUDT1
SCHEMBL26977882 0.76 ADORA2A (0.47) ADORA2AADORA1CSNK1A1CLK4NUDT1
SCHEMBL12985532 0.73 CHEK1 (0.39) CHEK1CHEK2HRH3CHRNB2CHRNA4
SCHEMBL16669652 0.73 FGFR4 (0.42) CHRNB2CHRNA4
SCHEMBL29314144 0.71 ADORA2A (0.38) ADORA2AADORA1CSNK1A1CLK4NUDT1
SCHEMBL2552574 0.70 SLC6A4 (0.44) CHEK1CHEK2HTR7
SCHEMBL25598905 0.69 ADORA2A (0.47) ADORA2AADORA1CSNK1A1CLK4NUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116635390-A Potent and selective compounds as serotonin 1B receptor modulators 莱科斯生物技术公司 2023-08-22 CN disclosed
EP-4225753-A1 POTENT AND SELCTIVE COMPOUNDS AS SEROTONIN 1B RECEPTOR MODULATORS Leukos Biotech, S.L. (ES) 2023-08-16 EP disclosed
WO-2022074103-A1 POTENT AND SELCTIVE COMPOUNDS AS SEROTONIN 1B RECEPTOR MODULATORS LEUKOS BIOTECH, S.L. (ES) 2022-04-14 WO disclosed