Colfenamate

Colfenamate

SCHEMBL29462552

NC(=O)COC(=O)c1ccccc1Nc1cccc(C(F)(F)F)c1

nearest known ligand 0.68

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.68
CYP1A2 P05177 1/20 0.68
CYP2C9 P11712 1/20 0.68
CYP2C19 P33261 1/20 0.68
YAP1 P46937 1/20 0.62
TEAD4 Q15561 1/20 0.62
TEAD2 Q15562 1/20 0.62
RXFP1 Q9HBX9 5/20 0.61
SIRT2 Q8IXJ6 2/20 0.55
ALDH1A1 P00352 1/20 0.52
GAA P10253 1/20 0.52
MAPT P10636 1/20 0.52
RAB9A P51151 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
MPO P05164 3/20 0.51
NTRK1 P04629 1/20 0.49
NTRK2 Q16620 1/20 0.49
KIF11 P52732 1/20 0.49
AKR1C3 P42330 1/20 0.48
AKR1C2 P52895 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Colfenamate SCHEMBL2110641 1.00 LMNA (0.68) LMNACYP1A2CYP2C9CYP2C19YAP1
SCHEMBL10597386 0.86 LMNA (0.71) LMNACYP1A2CYP2C9CYP2C19YAP1
SCHEMBL12715082 0.85 LMNA (0.91) LMNACYP1A2CYP2C9CYP2C19YAP1
SCHEMBL13299181 0.83 LMNA (0.67) LMNACYP1A2CYP2C9CYP2C19YAP1
SCHEMBL11494752 0.83 LMNA (0.67) LMNACYP1A2CYP2C9CYP2C19YAP1
SCHEMBL9271694 0.83 RXFP1 (0.70) LMNACYP1A2CYP2C9CYP2C19YAP1
SCHEMBL9270625 0.82 RXFP1 (0.73) LMNACYP1A2CYP2C9CYP2C19YAP1
Ufenamate SCHEMBL36095 0.82 CYP1A2 (0.72) LMNACYP1A2CYP2C9CYP2C19YAP1
SCHEMBL11520753 0.82 LMNA (0.66) LMNACYP1A2CYP2C9CYP2C19YAP1
Ufenamate SCHEMBL29376700 0.82 CYP1A2 (0.72) LMNACYP1A2CYP2C9CYP2C19YAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12226484-B2 Compositions having improved bioavailability of therapeutics TRx Biosciences Limited (GB) 2025-02-18 US disclosed
CN-115066291-B Aqueous capsule suspension concentrate based on polyurea shell material containing multifunctional aminocarboxylate 拜耳公司 2024-12-13 CN disclosed
CN-118317956-A Bis (hetero) aryl thioether oxadiazines as fungicidal compounds 拜耳公司 2024-07-09 CN disclosed
US-20240075147-A1 Compositions Having Improved Bioavailability of Therapeutics TRx Biosciences Limited (GB) 2024-03-07 US disclosed
EP-4312978-A2 COMPOSITIONS HAVING IMPROVED BIOAVAILABILITY OF THERAPEUTICS TRX Biosciences Limited (GB) 2024-02-07 EP disclosed
CN-111741945-B Crystalline forms 先正达参股股份有限公司 2024-01-09 CN disclosed
CN-110505874-B Molecules having pesticidal utility, and intermediates, compositions and methods related thereto 科迪华农业科技有限责任公司 2023-09-26 CN disclosed
WO-2022207580-A2 COMPOSITIONS HAVING IMPROVED BIOAVAILABILITY OF THERAPEUTICS TRx Biosciences Limited (GB) 2022-10-06 WO disclosed
CN-115135384-A Benzimidazole compound or its salt, and agricultural and horticultural insecticide and acaricide containing the same and method of using the same 日本农药株式会社 2022-09-30 CN disclosed
US-20220305125-A1 Compositions Having Improved Bioavailability of Therapeutics TRx Biosciences Limited (GB) 2022-09-29 US disclosed
CN-110461839-B JAK inhibitors containing 4-membered heterocyclic amides 施万生物制药研发IP有限责任公司 2022-08-23 CN disclosed
CN-110121500-B 4H-pyrrolopyridine compound or salt thereof, agricultural or horticultural insecticide containing same, and method for using same 日本农药株式会社 2022-05-03 CN disclosed
CN-110868861-B Agricultural compositions 萨卡帕·瓦达卡库塔 2022-03-15 CN disclosed